Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 99 hits in this display
BDBM59229(Pyrazolopyrimidone analog, RGB-286331)
BDBM59228(Pyrazolopyrimidone analog, RGB-285940)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM6027(N-(4-{[3-Ethyl-4-oxo-1-(2,4,6-trichlorophenyl)-4,5...)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM6025(3-Ethyl-6-(3-hydroxybenzyl)-1-(2,4,6-trichlorophen...)IC50: 14nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM6011(6-(4-Aminobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)
BDBM6012(3-Ethyl-6-(4-methoxybenzyl)-1-(2,4,6-trichlorophen...)IC50: 16nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6013(3-Ethyl-6-(4-hydroxybenzyl)-1-(2,4,6-trichlorophen...)IC50: 16nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6009(3-Ethyl-6-(pyrid-3-ylmethyl)-1-(2,4,6-trichlorophe...)IC50: 17nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6023(3-Ethyl-6-(3-hydroxy-4-methoxybenzyl)-1-(2,4,6-tri...)
BDBM6004(6-(3-Amino-2-methylbenzyl)-3-ethyl-1-(2,4,6-trichl...)
BDBM6021(6-(3,4-Dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)IC50: 20nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6022(6-(3,5-Dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)IC50: 22nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59235(PEGylated derivative, RGB-286276)IC50: 22nMAssay Description:In vitro kinase activity of PEGylated pyrazolopyrimidone CDK inhibitor or a 5 PEG-amine was coupled to ReactiGel agarose beads (Pierce, No. 20259).More data for this Ligand-Target Pair
BDBM6015(6-(4-(N,N-Dimethylamino)benzyl)-3-ethyl-1-(2,4,6-t...)IC50: 23nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6024(3-Ethyl-6-(3-hydroxy-4-methylbenzyl)-1-(2,4,6-tric...)IC50: 23nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6023(3-Ethyl-6-(3-hydroxy-4-methoxybenzyl)-1-(2,4,6-tri...)
IC50: 24nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM5998(6-Benzyl-3-ethyl-1-(2,4,6-trichlorophenyl)-4,5-dih...)IC50: 24nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6018(3-Ethyl-6-(4-hydroxy-3-methylbenzyl)-1-(2,4,6-tric...)IC50: 27nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6002(3-Ethyl-6-(2-(hydroxymethyl)benzyl)-1-(2,4,6-trich...)IC50: 27nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6007(3-Ethyl-6-(3-methoxybenzyl)-1-(2,4,6-trichlorophen...)IC50: 32nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59235(PEGylated derivative, RGB-286276)
BDBM6010(3-Ethyl-6-(pyrid-4-ylmethyl)-1-(2,4,6-trichlorophe...)IC50: 38nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6027(N-(4-{[3-Ethyl-4-oxo-1-(2,4,6-trichlorophenyl)-4,5...)
BDBM6005(3-Ethyl-6-(3-methylbenzyl)-1-(2,4,6-trichloropheny...)IC50: 39nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6008(6-(3-Aminobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)IC50: 40nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59229(Pyrazolopyrimidone analog, RGB-286331)
BDBM6021(6-(3,4-Dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)
IC50: 44nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM6014(6-(4-Bromobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)IC50: 58nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6022(6-(3,5-Dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)
IC50: 59nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6016(3-Ethyl-6-(4-methoxy-3-methylbenzyl)-1-(2,4,6-tric...)IC50: 67nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6025(3-Ethyl-6-(3-hydroxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 68nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM6019(3-Ethyl-6-(4-hydroxy-3-methoxybenzyl)-1-(2,4,6-tri...)IC50: 76nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59235(PEGylated derivative, RGB-286276)
IC50: 84nMAssay Description:In vitro kinase activity of PEGylated pyrazolopyrimidone CDK inhibitor or a 5 PEG-amine was coupled to ReactiGel agarose beads (Pierce, No. 20259).More data for this Ligand-Target Pair
BDBM6024(3-Ethyl-6-(3-hydroxy-4-methylbenzyl)-1-(2,4,6-tric...)
IC50: 88nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6013(3-Ethyl-6-(4-hydroxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 100nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6000(3-Ethyl-6-(2-methoxybenzyl)-1-(2,4,6-trichlorophen...)IC50: 100nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6020(6-(3,4-Dimethoxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)IC50: 110nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6017(3-Ethyl-6-(3-methoxy-4-methylbenzyl)-1-(2,4,6-tric...)IC50: 110nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6001(3-Ethyl-6-(2-hydroxybenzyl)-1-(2,4,6-trichlorophen...)IC50: 120nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6011(6-(4-Aminobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)
IC50: 150nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6012(3-Ethyl-6-(4-methoxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 150nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6025(3-Ethyl-6-(3-hydroxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 190nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6023(3-Ethyl-6-(3-hydroxy-4-methoxybenzyl)-1-(2,4,6-tri...)
IC50: 200nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59229(Pyrazolopyrimidone analog, RGB-286331)
BDBM6009(3-Ethyl-6-(pyrid-3-ylmethyl)-1-(2,4,6-trichlorophe...)
IC50: 220nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59228(Pyrazolopyrimidone analog, RGB-285940)
BDBM6021(6-(3,4-Dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)
IC50: 240nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6015(6-(4-(N,N-Dimethylamino)benzyl)-3-ethyl-1-(2,4,6-t...)
IC50: >260nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM5998(6-Benzyl-3-ethyl-1-(2,4,6-trichlorophenyl)-4,5-dih...)
IC50: 260nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6004(6-(3-Amino-2-methylbenzyl)-3-ethyl-1-(2,4,6-trichl...)
IC50: >270nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6008(6-(3-Aminobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)
IC50: 270nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6018(3-Ethyl-6-(4-hydroxy-3-methylbenzyl)-1-(2,4,6-tric...)
IC50: >270nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6002(3-Ethyl-6-(2-(hydroxymethyl)benzyl)-1-(2,4,6-trich...)
IC50: >270nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59228(Pyrazolopyrimidone analog, RGB-285940)
BDBM6007(3-Ethyl-6-(3-methoxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 410nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6010(3-Ethyl-6-(pyrid-4-ylmethyl)-1-(2,4,6-trichlorophe...)
IC50: 490nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6020(6-(3,4-Dimethoxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)
IC50: >510nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6024(3-Ethyl-6-(3-hydroxy-4-methylbenzyl)-1-(2,4,6-tric...)
IC50: 520nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6005(3-Ethyl-6-(3-methylbenzyl)-1-(2,4,6-trichloropheny...)
IC50: >560nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59227(Pyrazolopyrimidone analog, RGB-286147)
BDBM59228(Pyrazolopyrimidone analog, RGB-285940)
BDBM6019(3-Ethyl-6-(4-hydroxy-3-methoxybenzyl)-1-(2,4,6-tri...)
IC50: 860nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6016(3-Ethyl-6-(4-methoxy-3-methylbenzyl)-1-(2,4,6-tric...)
IC50: 870nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59235(PEGylated derivative, RGB-286276)
IC50: 890nMAssay Description:In vitro kinase activity of PEGylated pyrazolopyrimidone CDK inhibitor or a 5 PEG-amine was coupled to ReactiGel agarose beads (Pierce, No. 20259).More data for this Ligand-Target Pair
BDBM6014(6-(4-Bromobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)
IC50: >1.20E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6009(3-Ethyl-6-(pyrid-3-ylmethyl)-1-(2,4,6-trichlorophe...)
IC50: 1.30E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6027(N-(4-{[3-Ethyl-4-oxo-1-(2,4,6-trichlorophenyl)-4,5...)
IC50: 1.30E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6013(3-Ethyl-6-(4-hydroxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 2.00E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6015(6-(4-(N,N-Dimethylamino)benzyl)-3-ethyl-1-(2,4,6-t...)
IC50: >2.10E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6016(3-Ethyl-6-(4-methoxy-3-methylbenzyl)-1-(2,4,6-tric...)
IC50: >2.10E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6017(3-Ethyl-6-(3-methoxy-4-methylbenzyl)-1-(2,4,6-tric...)
IC50: 2.10E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6012(3-Ethyl-6-(4-methoxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 2.20E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6005(3-Ethyl-6-(3-methylbenzyl)-1-(2,4,6-trichloropheny...)
IC50: >2.20E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6004(6-(3-Amino-2-methylbenzyl)-3-ethyl-1-(2,4,6-trichl...)
IC50: >2.20E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6018(3-Ethyl-6-(4-hydroxy-3-methylbenzyl)-1-(2,4,6-tric...)
IC50: >2.20E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6011(6-(4-Aminobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)
IC50: 2.70E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6002(3-Ethyl-6-(2-(hydroxymethyl)benzyl)-1-(2,4,6-trich...)
IC50: 2.90E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6008(6-(3-Aminobenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl...)
IC50: 2.90E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM5998(6-Benzyl-3-ethyl-1-(2,4,6-trichlorophenyl)-4,5-dih...)
IC50: 3.00E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6010(3-Ethyl-6-(pyrid-4-ylmethyl)-1-(2,4,6-trichlorophe...)
IC50: 3.00E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6020(6-(3,4-Dimethoxybenzyl)-3-ethyl-1-(2,4,6-trichloro...)
IC50: 4.50E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6007(3-Ethyl-6-(3-methoxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: 5.00E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6019(3-Ethyl-6-(4-hydroxy-3-methoxybenzyl)-1-(2,4,6-tri...)
IC50: 6.60E+3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM59234(Pyrazolopyrimidone analog, RGB-310591)
BDBM6001(3-Ethyl-6-(2-hydroxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: >1.10E+4nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
BDBM6000(3-Ethyl-6-(2-methoxybenzyl)-1-(2,4,6-trichlorophen...)
IC50: >2.20E+4nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
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