Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM7615(2,4-bis anilino pyrimidine deriv. 11 | 4-N-(2,5-di...)
IC50: 800nMAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7597(4,6-bis anilino pyrimidine deriv. 10 | 4-N-(2,5-di...)
IC50: 1.00E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7615(2,4-bis anilino pyrimidine deriv. 11 | 4-N-(2,5-di...)
IC50: 1.00E+3nMAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7607(2,4-bis anilino pyrimidine deriv. 3 | 4-N-(2-chlor...)
IC50: 1.00E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7615(2,4-bis anilino pyrimidine deriv. 11 | 4-N-(2,5-di...)
BDBM7611(2,4-bis anilino pyrimidine deriv. 7 | 4-N-(3-chlor...)
IC50: 2.00E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7611(2,4-bis anilino pyrimidine deriv. 7 | 4-N-(3-chlor...)
IC50: 5.00E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7607(2,4-bis anilino pyrimidine deriv. 3 | 4-N-(2-chlor...)
IC50: 6.00E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
BDBM7597(4,6-bis anilino pyrimidine deriv. 10 | 4-N-(2,5-di...)
IC50: 2.20E+4nMAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair