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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
222
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Target
Sigma non-opioid intracellular receptor 1
(Mus musculus (Mouse))
Soochow University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 2.90nM
Assay Description:
Inhibition of radioligand binding to sigma1 receptor in C57BL/6 mouse brain membranes
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Target
Sigma non-opioid intracellular receptor 1
(Homo sapiens (Human))
Medical College Of Georgia
Curated by
PDSP K
i
Database
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Ki: 8.70nM
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 12nM
Assay Description:
Irreversible inhibition of recombinant human MAO-A expressed in baculovirus infected BT1 cells using p-tyramine as substrate by Lineweaver-Burk plot ...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 40nM
Assay Description:
Reversible inhibition of recombinant human MAOA expressed in Pichia pastoris using varying levels of kynuramine as substrate measured after 5 mins by...
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Target
Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 54nM
Assay Description:
Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...
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Target
Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
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Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 54nM
Assay Description:
Inhibitory activity against monoamine oxidase A in isolated bovine brain mitochondria
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Target
Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
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Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 54nM ΔG°: -43.3kJ/mole
pH: 7.4 T: 2°C
Assay Description:
MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...
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Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 54nM
Assay Description:
Inhibition of bovine brain mitochondrial MAO-A by fluorometric assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 220nM
Assay Description:
Irreversible inhibition of recombinant human MAOA expressed in Pichia pastoris using varying levels of kynuramine as substrate measured after 5 mins ...
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Target
Sigma intracellular receptor 2
(Mus musculus (Mouse))
Soochow University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 505nM
Assay Description:
Inhibition of radioligand binding to sigma2 receptor in C57BL/6 mouse brain membranes
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University Of Turku
Curated by
PDSP K
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BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Ki: 1.00E+3nM
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University Of Turku
Curated by
PDSP K
i
Database
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BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Ki: 1.00E+3nM
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 1.20E+3nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate after 60 mins by Lineweaver-Burk plot
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Target
Cytochrome P450 2B1
(Rattus norvegicus)
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 1.50E+3nM
Assay Description:
Mechanism based inhibition of rat cytochrome P450 CYP2B1 measured by 7-EFC O-deethylation activity
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 5.60E+3nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate after 60 mins by Lineweaver-Burk plot
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 5.80E+4nM
Assay Description:
Inhibition of bovine brain mitochondrial MAO-B by fluorometric assay
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 5.80E+4nM
Assay Description:
Inhibition of bovine brain MAOB using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 5.80E+4nM
Assay Description:
MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
Ki: 5.80E+4nM
Assay Description:
Inhibitory activity against monoamine oxidase B in isolated bovine brain mitochondria
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 0.00490nM
Assay Description:
Inhibition of human monoamine oxidase A
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 0.420nM
Assay Description:
Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assay
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 0.5nM
Assay Description:
Inhibition of MAO-B in rat whole brain homogenate in presence of clorgyline
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 0.5nM
Assay Description:
The compounds of the present invention obtained in the Production Examples were examined for the inhibitory effect on human monoamineoxydase enzymes ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 0.610nM
Assay Description:
Inhibition of human full length recombinant MAO-A expressed in insect cells using kynuramine as substrate
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Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 0.700nM
Assay Description:
In vitro Inhibitory activity of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT (serotonin)
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1nM
Assay Description:
Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1nM
Assay Description:
Inhibition of MAO-A (unknown origin) expressed in mouse GL26 cells using 14C 5-hydroxytryptamine as substrate pre-incubated for 20 mins followed by s...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.10nM
Assay Description:
Inhibition of MAO-A (unknown origin)
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.20nM
Assay Description:
Inhibition of MAO-A (unknown origin)
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.60nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in Sf9 cells using p-tyramine as substrate preincubated for 15 mins followed by substrate addition fo...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 2nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells using tyramine as substrate preincubated for 1 hr f...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.20nM
Assay Description:
Inhibition of recombinant human MAO-B
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.5nM
Assay Description:
Inhibition of recombinant human MAOA using kynuramine as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.5nM
Assay Description:
Inhibition of human recombinant MAOA expressed in microsomes of baculovirus-infected insect cell using kynuramine as substrate preincubated for 20 mi...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 2.5nM
Assay Description:
Inhibition of human recombinant MAOA expressed in microsomes of baculovirus-infected insect cell using kynuramine as substrate preincubated for 20 mi...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.60nM
Assay Description:
Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometry
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.60nM
Assay Description:
Inhibition of human recombinant MAOA expressed in insect cell microsomes using kynuramine as substrate after 20 mins by fluorescence spectrophotometr...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of human recombinant MAO-A by multimode plate reader assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of human microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in 4-hydroxyquinoline formation using...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of recombinant human MAO-A using kynuramine as substrate after 30 mins by fluorescence assay
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 30 mins by fluorescence ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate incubated for 30 mins by fluor...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 30 mins by fluorimetric ...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected High 5 insect cells using kynuramine as substrate incubated for 30 mins by sp...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of human recombinant MAO-A using kynuramine as substrate measured after 30 mins by fluorescence assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.70nM
Assay Description:
Inhibition of human recombinant MAO-A using kynuramine as substrate after 30 mins by fluorescence spectrophotometry
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.90nM
Assay Description:
Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate addition
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 2.90nM
Assay Description:
Inhibition of recombinant human MAOA expressed in baculovirus infected in BTI cells using kynuramine as substrate after 30 mins by fluorescence based...
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Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.90nM
Assay Description:
Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3nM
Assay Description:
Inhibition of human recombinant MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.10nM
Assay Description:
Inhibition of MAO-A (unknown origin) using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazolecarboxylic acid as substrate by MAO-Glo assay
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Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 3.10nM
Assay Description:
Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.10nM
Assay Description:
Inhibition of MAO-A (unknown origin)
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 3.10nM
Assay Description:
Inhibition of MAOA by spectrophotometry
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Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.10nM
Assay Description:
Inhibition of bovine brain mitochondria MAO-A by spectrofluorimetry
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.20nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI-TN- 5B1-4 insect cells using kynuramine as substrate preincubated for 10 ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.40nM
Assay Description:
Inhibition of recombinant human MAO-A using kynuramine as substrate after 30 mins by fluorescence method
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 3.40nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 30 mins by fluorescence ...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 3.40nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus-infected insect cells using p-tyramine as substrate preincubated for 15 min...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 3.40nM
Assay Description:
Inhibition of recombinant human microsomal MAOA expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 15 ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.40nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells using p-tyramine as substrate preincubated for 15 m...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.60nM
Assay Description:
Inhibition of TNF-alpha release was determined in LPS-stimulated human whole blood assay
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Amine oxidase [flavin-containing] A
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.70nM
Assay Description:
Inhibition of MAO-A in bovine brain mitochondria using serotonin as substrate preincubated for 30 mins measured after 30 mins by spectrofluorimetric ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 3.80nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected insect cell microsomes using kynuramine as substrate measured after 30 mins b...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in BTI-TN-5B1-4 cells by para-tyramine oxidation assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4nM
Assay Description:
Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.10nM
Assay Description:
Inhibition of recombinant human MAO-A using p-tyramine substrate preincubated for 15 mins before substrate addition measured after 20 mins by fluores...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.10nM
Assay Description:
Inhibition of human recombinant MAOA assessed as H2O2 production by Amplex Red reagent-based assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.10nM
Assay Description:
Inhibition of human recombinant MAO-A using p-tyramine as substrate incubated for 15 mins prior to substrate addition measured after 20 mins by fluor...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.40nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in production of H202 usi...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected insect BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-t...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected BTI insect cells assessed as hydrogen peroxide production after 15 mins by Amp...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human recombinant MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human MAOA by fluorimetry
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human recombinant MAOA by fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate incubated for 15 mins prior to substrate...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.46nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect sells assessed as hydrogen peroxide production by fluorim...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus-infected insect BTI-TN-5B1-4 cells assessed as p-tyramine conversion to H2O...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human microsomal MAO-A expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O2 production...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BT1-TN-5B1-4 cells assessed as inhibition of production of hydrogen peroxide ...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate assessed as reduc...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus-infected BTI-TN-5B1-4 cell microsomes assessed as decrease in H2O2 production using p-...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 cells
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of recombinant human MAO-A using kynuramine as substrate after 20 mins by fluorescence assay
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.5nM
pH: 7.4 T: 2°C
Assay Description:
The effects of the test compounds on hMAO isoform enzymatic activity were evaluated by measuring their effects on the production of hydrogen peroxide...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.5nM
pH: 7.4
Assay Description:
The assay was performed in a polystyrene 96-well plate having flat bottom containing 200 μL of the total reaction mixture. For each assay, mixtu...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as inhibition of hydrogen peroxide product...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of recombinant human MAOA expressed in baculovirus infected BTI insect cells using p-tyramine as substrate measured after 15 mins by Ample...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.70nM
Assay Description:
Inhibition of human MAO-A expressed in baculovirus infected BTI insect cells preincubated for 15 mins
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.90nM
Assay Description:
Inhibition of human recombinant MAO-A using pargyline as incubated for 20 mins measuring increase in emission signal at 310 nm multimode plate reader...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.90nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.90nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells preincubated for 10 mins followed by addition of kynuramine ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 4.90nM
Assay Description:
Inhibition of human recombinant MAO-A using kynuramine substrate by spectrophotometric assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 5nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 5.20nM
Assay Description:
Inhibition of human recombinant MAO-A assessed as inhibition of production of hydrogen peroxide after 15 mins by Amplex Red fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 5.40nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using tyramine as substrate pretreated for 30 mins followed ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.20nM
Assay Description:
Inhibition of human recombinant MAOA using kynuramine as substrate preincubated for 30 mins followed by substrate addition
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.70nM
Assay Description:
Inhibition of human recombinant MAO-A using kynuramine as substrate preincubated with compound for 15 mins measured after 20 mins by fluorometric ana...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 7.90nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate measured after 30 mins by fluo...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 7.90nM
pH: 7.4
Assay Description:
Recombinant human MAO-A and MAO-B (5 mg/mL) were purchased from Sigma-Aldrich, pre-aliquoted and stored at -80 °C. Solutions of test compounds we...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 7.90nM
Assay Description:
Inhibition of recombinant human MAO-A using kynuramine as substrate after 30 mins by fluorescence assay
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 8nM
Assay Description:
Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 8nM
Assay Description:
Inhibition of recombinant human MAOA using p-tyramine as substrate after 30 mins by Amplex red based spectrophotometric analysis
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8nM
Assay Description:
Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins by...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 10nM
Assay Description:
Reversible inhibition of recombinant human MAO-A assessed as residual activity using kynuramine as substrate preincubated for 30 mins followed by dia...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: <10nM
Assay Description:
Inhibition of recombinant human MAO-A using kynuramine as substrate after 20 mins by fluorescence assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 12nM
Assay Description:
Inhibition of human MAOA after 1 hr by luminescence assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 13nM
Assay Description:
Inhibition of recombinant human MAOA using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured after 15 mins by ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 16nM
Assay Description:
Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAO-A preincubated for 30 mins followed by p-tyramine hydrochloride addition measured after 30 mins by Amplex red flu...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 21nM
Assay Description:
Inhibition of human MAO-A
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 25nM
Assay Description:
Inhibition of human recombinant MAOA using kynuramine as substrate incubated for 10 mins by UPLC-ESI-MS/MS analysis
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 27nM
Assay Description:
Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 30nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate using [14C]-5HT as substrate preincubated for 30 mins followed by substrate addition measured after 20 mi...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 30.2nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assay
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 38nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in insect cells using p-tyramine as substrate preincubated for 30 mins followed by substrate addition...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 40nM
Assay Description:
Inhibition of recombinant human MAOA expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 30 mins follow...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 43nM
Assay Description:
Inhibition of human MAO-A using p-tyramine as substrate by fluorimetric analysis
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 48nM
Assay Description:
Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 50nM
Assay Description:
Inhibition of human MAO-A preincubated for 5 mins followed by addition of Kynuramine substrate and measured after 30 mins by plate reader method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 189nM
Assay Description:
Inhibition of recombinant human microsomal MAO-A expressed in baculovirus-infected insect cells using p-tyramine as substrate assessed as H2O2 produc...
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 189nM
Assay Description:
Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 260nM
Assay Description:
Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assay
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Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 680nM
Assay Description:
In vitro Inhibitory activity of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA (phenethylamine)
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: >1.00E+3nM
Assay Description:
Inhibition of recombinant human MAOB using benzylamine as substrate after 30 mins by Amplex red based spectrophotometric analysis
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: >1.00E+3nM
Assay Description:
Inhibition of recombinant human MAO-B using benzylamine as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins b...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.90E+3nM
Assay Description:
In vitro inhibitory activity on rat brain by monoamine oxidase A (MAO-A)
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.90E+3nM
Assay Description:
In vitro inhibitory activity on rat brain MAO-B.
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI insect cells using benzylamine as substrate after 30 mins by spectrophoto...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells preincubated for 10 mins followed by addition of benzylamine...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of human recombinant MAOB using benzylamine as substrate preincubated for 30 mins followed by substrate addition
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.05E+3nM
Assay Description:
Inhibition of MAOA in rat liver homogenates preincubated for 60 mins
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.05E+3nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate after 60 mins by residual activity plot
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.21E+3nM
Assay Description:
Inhibition of human microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in 4-hydroxyquinoline formation using...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.21E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI-TN- 5B1-4 insect cells using kynuramine as substrate preincubated for 10 ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.34E+3nM
Assay Description:
Inhibition of recombinant human MAOB expressed in baculovirus infected in BTI cells using kynuramine as substrate after 30 mins by fluorescence based...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.43E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 30 mins by fluorimetric ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.50E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected insect cell microsomes using kynuramine as substrate measured after 30 mins b...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.55E+3nM
Assay Description:
Inhibition of human recombinant MAOB expressed in microsomes of baculovirus-infected insect cell using kynuramine as substrate preincubated for 20 mi...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.55E+3nM
Assay Description:
Inhibition of human recombinant MAOB expressed in microsomes of baculovirus-infected insect cell using kynuramine as substrate preincubated for 20 mi...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.72E+3nM
Assay Description:
Inhibition of recombinant human MAOA using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additio...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.72E+3nM
Assay Description:
Inhibition of rat liver MAOA after 60 mins pre-incubation
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.76E+3nM
Assay Description:
Inhibition of human recombinant MAO-A using p-tyramine as substrate assessed as production of H2O2 incubated for 15 mins prior to substrate addition ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 3.20E+3nM
Assay Description:
Inhibition of recombinant human MAOA using kynuramine as substrate measured for 30 mins by fluorescence spectrophotometric assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.19E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate incubated for 30 mins by fluor...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.19E+3nM
Assay Description:
Inhibition of human recombinant MAO-B using kynuramine as substrate measured after 30 mins by fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.19E+3nM
Assay Description:
Inhibition of human recombinant MAO-B using kynuramine as substrate after 30 mins by fluorescence spectrophotometry
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.19E+3nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 30 mins by fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.19E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected High 5 insect cells using kynuramine as substrate incubated for 30 mins by sp...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.46E+3nM
Assay Description:
Inhibition of human recombinant MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.46E+3nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramin...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 5.02E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 30 mins by fluorescence ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 5.02E+3nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 30 mins by fluorescence method
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 5.80E+3nM
Assay Description:
Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins measuring increase in emission signal at 400 nm multimode p...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 7.65E+3nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells using benzylamine as substrate preincubated for 1 h...
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 8.00E+3nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate using [14C]-phenylethylamine as substrate preincubated for 30 mins followed by substrate addition measure...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 8.85E+3nM
pH: 7.4
Assay Description:
Recombinant human MAO-A and MAO-B (5 mg/mL) were purchased from Sigma-Aldrich, pre-aliquoted and stored at -80 °C. Solutions of test compounds we...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 8.85E+3nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 30 mins by fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 8.85E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate measured after 30 mins by fluo...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 8.87E+3nM
Assay Description:
Inhibition of human recombinant MAO-B incubated for 30 mins by fluorescence based assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.10E+4nM
Assay Description:
Inhibition of human recombinant MAO-B using kynuramine substrate by spectrophotometric assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.36E+4nM
Assay Description:
Inhibition of recombinant human microsomal MAOB expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 15 ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.36E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in baculovirus-infected insect cells using p-tyramine as substrate preincubated for 15 min...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 1.36E+4nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells using p-tyramine as substrate preincubated for 15 m...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.42E+4nM
Assay Description:
Inhibition of recombinant human MAOB using kynuramine as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 1.43E+4nM
Assay Description:
Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.03E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect cells using p-tyramine as substrate preincubated for 30 mins followed by substrate addition...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.03E+4nM
Assay Description:
Inhibition of human MAO-B
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.03E+4nM
Assay Description:
Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 30 mins follow...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 2.08E+4nM
Assay Description:
Inhibition of human recombinant MAO-B by multimode plate reader assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 2.08E+4nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 30 mins by fluorescence ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Padova
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 2.26E+4nM
Assay Description:
Inhibition of recombinant human MAO-A
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Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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IC50: 5.00E+4nM
Assay Description:
Inhibitory activity against rat brain mitochondrial Monoamine oxidase
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 5.43E+4nM
Assay Description:
Inhibition of human recombinant MAOB
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: >6.00E+4nM
Assay Description:
Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >6.00E+4nM
Assay Description:
Inhibition of recombinant human MAOB using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additio...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as inhibition of hydrogen peroxide product...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramin...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI insect cells assessed as hydrogen peroxide production after 15 mins by Amp...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human MAOB by fluorimetry
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells by para-tyramine oxidation assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate assessed as reduc...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB by fluorimetric method
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected insect BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-t...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect sells assessed as hydrogen peroxide production by fluorim...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus-infected BTI-TN-5B1-4 cell microsomes assessed as decrease in H2O2 production using p-...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
pH: 7.4
Assay Description:
The assay was performed in a polystyrene 96-well plate having flat bottom containing 200 μL of the total reaction mixture. For each assay, mixtu...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in baculovirus-infected insect BTI-TN-5B1-4 cells assessed as p-tyramine conversion to H2O...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.14E+4nM
pH: 7.4 T: 2°C
Assay Description:
The effects of the test compounds on hMAO isoform enzymatic activity were evaluated by measuring their effects on the production of hydrogen peroxide...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 20 mins by fluorescence assay
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BT1-TN-5B1-4 cells assessed as inhibition of production of hydrogen peroxide ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate incubated for 15 mins prior to substrate...
More data for this Ligand-Target Pair
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.14E+4nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...
More data for this Ligand-Target Pair
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.17E+4nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 cells
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.20E+4nM
Assay Description:
Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cells using p-tyramine as substrate measured after 15 mins by Ample...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.34E+4nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decrease in H2O2...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.34E+4nM
Assay Description:
Inhibition of human recombinant MAO-B assessed as inhibition of production of hydrogen peroxide after 15 mins by the Amplex Red fluorimetric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.34E+4nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...
More data for this Ligand-Target Pair
Target Info
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.34E+4nM
Assay Description:
Inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O2 production...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 6.55E+4nM
Assay Description:
Inhibition of human recombinant MAO-B preincubated for 30 mins followed by p-tyramine hydrochloride addition measured after 30 mins by Amplex red flu...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.55E+4nM
Assay Description:
Inhibition of human recombinant MAOB using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 6.58E+4nM
Assay Description:
Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells preincubated for 15 mins
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 9.80E+4nM
Assay Description:
Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrate
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 9.80E+4nM
Assay Description:
Inhibition of bovine brain mitochondria MAO-B using benzylamine substrate after 60 mins by fluorimetric method
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.01E+5nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate after 60 mins by residual activity plot
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: 4.01E+5nM
Assay Description:
Inhibition of rat liver MAOB after 60 mins pre-incubation
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Hacettepe University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.01E+5nM
Assay Description:
Inhibition of MAOB in rat liver homogenates preincubated for 60 mins
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Acetylcholinesterase
(Homo sapiens (Human))
Okayama University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: >5.00E+5nM
Assay Description:
Inhibition of human recombinant AChE expressed in HEK293 cells using acetylthiocholine iodide as substrate preincubated for 30 mins followed by subst...
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Cholinesterase
(Homo sapiens (Human))
Okayama University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
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Affinity Data
IC50: >5.00E+5nM
Assay Description:
Inhibition of human recombinant BuChE expressed in HEK293 cells using S-butyrylthiocholine iodide as substrate preincubated for 30 mins followed by s...
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Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
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Affinity Data
IC50: 9.40E+5nM
Assay Description:
Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric method
More data for this Ligand-Target Pair
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.21E+6nM
Assay Description:
Inhibition of recombinant human MAOB using kynuramine as substrate measured for 30 mins by fluorescence spectrophotometric assay
More data for this Ligand-Target Pair
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Copy BDB DOI
Target
Amine oxidase [flavin-containing] B
(Bos taurus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.40E+6nM
Assay Description:
Inhibition of bovine brain mitochondria MAO-B by spectrofluorimetry
More data for this Ligand-Target Pair
Target Info
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM15581
(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.40E+6nM
Assay Description:
Inhibition of MAOB by spectrophotometry
More data for this Ligand-Target Pair
Target Info
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