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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetCholesterol side-chain cleavage enzyme, mitochondrial(Rattus norvegicus)
Lucknow University

Curated by ChEMBL
LigandPNGBDBM50476074(Gentamicin | SCH-9724 | Uromycine)
Affinity DataIC50:  445nMAssay Description:Antibacterial activity against Streptococcus faecalis by broth microdilution techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNH(3)-dependent NAD(+) synthetase(Bacillus subtilis)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50366389(GENTAMICIN)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against Bacillus subtilis NAD synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50366389(GENTAMICIN)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human DHFR after 2 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Bos taurus (Cattle))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50366389(GENTAMICIN)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of bovine DHFR after 2 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50011926(4-amino-2-[2,4-diamino-5-(3-amino-6-aminomethyl-4,...)
Affinity DataIC50:  7.90E+4nMAssay Description:in vitro inhibitory activity against Lysosomal phospholipase A1 consisting of negatively charged liposomes and lysosomal extracts. p<0.05More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University Of Athens

Curated by ChEMBL
LigandPNGBDBM50366389(GENTAMICIN)
Affinity DataIC50:  9.42E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed