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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
13
hits in this display
Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
University Of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
Ki: 1.20E+3nM
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
Ki: 2.00E+3nM
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Upr Centre
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
Ki: 2.30E+3nM
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Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
Ki: 2.70E+3nM
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
4-aminobutyrate aminotransferase, mitochondrial
(Sus scrofa)
TBA
Curated by
ChEMBL
Ligand
BDBM50280206
((2S)-2-amino-2-methyl-3-(phosphonooxy)propanoic ac...)
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Affinity Data
Ki: 5.70E+6nM
Assay Description:
Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminase
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Target
Bifunctional aspartokinase/homoserine dehydrogenase 1
(Escherichia coli)
University Of Akron
Ligand
BDBM93001
(O-phospho-L-serine)
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Affinity Data
Ki: 1.20E+7nM
Assay Description:
Analogues of L-aspartic acid and beta-aspartyl phosphate were examined as inhibitors in the aspartokinase I reaction by using the coupled reaction wi...
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Target
Glutamate carboxypeptidase 2 [44-750]
(Homo sapiens (Human))
Nci-Fcrdc
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
IC50: 5.23E+5nM
pH: 7.4 T: 2°C
Assay Description:
The inhibition concentration values of GCPII were determined using the radioenzymatic assay with [3H] NAAG (radiolabeled on the terminal glutamate). ...
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
EC50: 1.00E+3nM
Assay Description:
Agonistic activity at Metabotropic glutamate receptor 4 expressed in mammalian cells by GTPgammaS binding assay
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Target Info
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3D Structure (crystal)
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
EC50: 2.70E+3nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR6 in rat
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.30E+3nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR4a in human
More data for this Ligand-Target Pair
Target Info
PDB
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antibodypedia
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Ligand Info
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ChEBI
CHEMBL
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In Depth
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Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
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Affinity Data
EC50: 1.60E+5nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR7 in rat
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
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Ligand Info
Purchase
ChEBI
CHEMBL
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KEGG
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PC sid
PDB
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Upr Centre
Curated by
PDSP K
i
Database
Ligand
BDBM17664
((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 4.00E+3nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR4a in rat
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
DrugBank
KEGG
MMDB
PC cid
PC sid
PDB
Patents
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In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI