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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataKi:  2.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280206((2S)-2-amino-2-methyl-3-(phosphonooxy)propanoic ac...)
Affinity DataKi:  5.70E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBifunctional aspartokinase/homoserine dehydrogenase 1(Escherichia coli)
University Of Akron

LigandPNGBDBM93001(O-phospho-L-serine)
Affinity DataKi:  1.20E+7nMAssay Description:Analogues of L-aspartic acid and beta-aspartyl phosphate were examined as inhibitors in the aspartokinase I reaction by using the coupled reaction wi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2 [44-750](Homo sapiens (Human))
Nci-Fcrdc

LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataIC50:  5.23E+5nMpH: 7.4 T: 2°CAssay Description:The inhibition concentration values of GCPII were determined using the radioenzymatic assay with [3H] NAAG (radiolabeled on the terminal glutamate). ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic activity at Metabotropic glutamate receptor 4 expressed in mammalian cells by GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Cns Research

Curated by ChEMBL
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataEC50:  2.70E+3nMAssay Description:Concentration for half maximal activation of metabotropic glutamate mGluR6 in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataEC50:  1.30E+3nMAssay Description:Concentration for half maximal activation of metabotropic glutamate mGluR4a in humanMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Cns Research

Curated by ChEMBL
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataEC50:  1.60E+5nMAssay Description:Concentration for half maximal activation of metabotropic glutamate mGluR7 in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataEC50:  4.00E+3nMAssay Description:Concentration for half maximal activation of metabotropic glutamate mGluR4a in ratMore data for this Ligand-Target Pair