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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373036(CHEMBL259621)
Affinity DataKi:  450nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMast cell carboxypeptidase A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataKi:  450nMAssay Description:The compound was evaluated for the inhibition of Carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Bos taurus (bovine))
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataKi:  500nMAssay Description:Inhibition of bovine carboxypeptidase A1More data for this Ligand-Target Pair
TargetCarboxypeptidase B(Homo sapiens (Human))
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Helicoverpa zea (Corn earworm moth) (Heliothis zea...)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataKi:  1.19E+4nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Serratia marcescens)TBA
LigandPNGBDBM50488290(CHEMBL2283143)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of Pseudomonas aeruginosa IMP1 metallo-beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetMetallo-beta-lactamase type 2(Serratia marcescens)TBA
LigandPNGBDBM50488285((2R,3R)-2,3-DIBENZYLSUCCINIC ACID)
Affinity DataIC50:  210nMAssay Description:Inhibition of Pseudomonas aeruginosa IMP1 metallo-beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of purified Carboxypeptidase B (CPB) by clot lysis assay in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase M(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of purified Carboxypeptidase M (CPM) by clot lysis assay in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed