Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetTransthyretin(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50530238(1,4,7,10,13,16-Hexaoxacyclooctadecane | 1,4,7,10,1...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of ANS binding to TTR V30M mutant (unknown origin) expressed in Escherichia coli assessed as BC50 for ANS binding to TTR at 5 uM in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50530238(1,4,7,10,13,16-Hexaoxacyclooctadecane | 1,4,7,10,1...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of ANS binding to TTR V30M mutant (unknown origin) expressed in Escherichia coli assessed as BC50 for ANS binding to TTR at 5 uM in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50530238(1,4,7,10,13,16-Hexaoxacyclooctadecane | 1,4,7,10,1...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of ANS binding to TTR V30M mutant (unknown origin) expressed in Escherichia coli assessed as BC50 for ANS binding to TTR at 100 mM in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50530238(1,4,7,10,13,16-Hexaoxacyclooctadecane | 1,4,7,10,1...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of ANS binding to TTR V30M mutant (unknown origin) expressed in Escherichia coli assessed as BC50 for ANS binding to TTR at 100 mM in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed