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Found 114 Enz. Inhib. hit(s) with Target = 'ATP-binding cassette sub-family C member 8'
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118351((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50012957(1-((p-(2-(5-chloro-o-anisamido)ethyl)phenyl)sulfon...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human SUR1/Kir6.2 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50190500(6-chloro-3-(1-methyl-1-phenylethyl)amino-4H-thieno...)
Affinity DataIC50:  81nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cells in presence of 2 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50153520((S)-2-ethoxy-4-(2-(3-methyl-1-(2-(piperidin-1-yl)p...)
Affinity DataIC50:  106nMAssay Description:In vitro displacement of [3H]-glibenclamide (IC50=0.61) from COS-1 cells expressing Sulfonylurea receptor 1 (SUR-1)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118349((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50153521(2-Methoxy-4-{[(S)-3-methyl-1-(2-piperidin-1-yl-phe...)
Affinity DataIC50:  163nMAssay Description:In vitro displacement of [3H]-glibenclamide (IC50=0.61) from COS-1 cells expressing Sulfonylurea receptor 1 (SUR-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118348((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  180nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363009(CHEMBL1946412)
Affinity DataIC50:  200nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118360(CHEMBL336586 | tert-Butyl-(2-chloro-7,7-dioxo-4,7-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363013(CHEMBL191539)
Affinity DataIC50:  240nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363006(CHEMBL363989)
Affinity DataIC50:  280nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50153522(2-(2-Fluoro-ethoxy)-4-{[(S)-3-methyl-1-(2-piperidi...)
Affinity DataIC50:  281nMAssay Description:In vitro displacement of [3H]-glibenclamide (IC50=0.61) from COS-1 cells expressing Sulfonylurea receptor 1 (SUR-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataIC50:  286nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cells in presence of 2 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataIC50:  320nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118343((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  340nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363004(CHEMBL1946140)
Affinity DataIC50:  350nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50130735((7-Chloro-1,1-dioxo-1,4-dihydro-1lambda*6*-benzo[1...)
Affinity DataIC50:  480nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363007(CHEMBL1946272)
Affinity DataIC50:  520nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362998(CHEMBL1945810)
Affinity DataIC50:  620nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50023475(CHEMBL2111887)
Affinity DataIC50:  640nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363002(CHEMBL115565)
Affinity DataIC50:  760nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363003(CHEMBL1946139)
Affinity DataIC50:  1.41E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363008(CHEMBL1946410)
Affinity DataIC50:  1.67E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362992(CHEMBL1946411)
Affinity DataIC50:  1.73E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363011(CHEMBL189093)
Affinity DataIC50:  1.75E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362991(CHEMBL1946273)
Affinity DataIC50:  1.81E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363001(CHEMBL1946137)
Affinity DataIC50:  2.05E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118355((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363012(CHEMBL1946759)
Affinity DataIC50:  2.98E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362995(CHEMBL1945807)
Affinity DataIC50:  3.03E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362997(CHEMBL1945809)
Affinity DataIC50:  3.58E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362990(CHEMBL1946138)
Affinity DataIC50:  3.78E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363010(CHEMBL1946414)
Affinity DataIC50:  4.93E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362993(CHEMBL1944656)
Affinity DataIC50:  6.31E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50099573(1N-[4-methoxy-3-methylamino(thioxo)methylsulfamoyl...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of human SUR1/Kir6.2 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363005(CHEMBL1946270)
Affinity DataIC50:  8.67E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362994(CHEMBL1946760)
Affinity DataIC50: >1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362993(CHEMBL1944656)
Affinity DataIC50: >1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362992(CHEMBL1946411)
Affinity DataIC50: >1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362991(CHEMBL1946273)
Affinity DataIC50: >1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362990(CHEMBL1946138)
Affinity DataIC50: >1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118351((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50363000(CHEMBL1946136)
Affinity DataIC50:  2.65E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362999(CHEMBL1946134)
Affinity DataIC50:  3.75E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362996(CHEMBL1945808)
Affinity DataIC50:  3.89E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Rattus norvegicus)
Universit£ de Li£ge

Curated by ChEMBL
LigandPNGBDBM50362989(CHEMBL1945806)
Affinity DataIC50: >5.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118349((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  1.46E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataIC50:  1.65E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118343((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  1.87E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM86248(CAS_364-98-7 | NSC_3019 | diazoxide)
Affinity DataIC50:  1.94E+5nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cells in presence of 2 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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