Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'Complex of Sliding-clamp-loader large subunit [R175L] and Sliding-clamp-loader small subunit'
LigandPNGBDBM36324(6-nitro-indolyl- 2'-deoxyriboside triphosphate...)
Affinity DataKi:  5.00E+3nM ΔG°:  -30.3kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM36316(5-ethyl-indolyl- 2'-deoxyriboside triphosphate...)
Affinity DataKi:  1.10E+4nM ΔG°:  -28.3kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM36319(5-nitro-indolyl- 2'-deoxyriboside triphosphate...)
Affinity DataKi:  1.64E+4nM ΔG°:  -27.3kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM36312(ATP{gamma}S | adenosine 5'-O-(3-thiotriphospha...)
Affinity DataKi:  3.32E+4nM ΔG°:  -25.6kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM36317(5-ethylene-indolyl- 2'-deoxyriboside triphosph...)
Affinity DataKi:  3.40E+4nM ΔG°:  -25.5kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM36323(4-nitro-indolyl- 2'-deoxyriboside triphosphate...)
Affinity DataKi:  4.16E+4nM ΔG°:  -25.0kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM36318(5-carboxylate-indolyl- 2'-deoxyriboside tripho...)
Affinity DataKi: <2.00E+5nM ΔG°: <-21.1kJ/molepH: 7.5 T: 2°CAssay Description:ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed