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Found 4 Enz. Inhib. hit(s) with Target = 'Efflux pump membrane transporter'
TargetEfflux pump membrane transporter(Escherichia coli)
University Of Oklahoma

LigandPNGBDBM81507(MC-207,110)
Affinity DataKd:  1.10E+5nMpH: 6.0Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEfflux pump membrane transporter(Escherichia coli)
University Of Oklahoma

LigandPNGBDBM50336500((E)-N-(9-(2-(ethoxycarbonyl)phenyl)-6-(ethylamino)...)
Affinity DataKd:  1.03E+4nMpH: 8.4Assay Description:Binding affinity to Escherichia coli K-12 multidrug efflux protein AcrB at pH 8.4 by equilibrium dialysis methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEfflux pump membrane transporter(Escherichia coli)
University Of Oklahoma

LigandPNGBDBM282((3R,4S,5R,6R)-5-hydroxy-6-[(2-hydroxy-3-{[4-hydrox...)
Affinity DataKd:  5.30E+5nMpH: 7.5Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEfflux pump membrane transporter(Escherichia coli)
University Of Oklahoma

LigandPNGBDBM81507(MC-207,110)
Affinity DataKd:  5.90E+5nMpH: 7.5Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed