Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with Target = 'Adenosine transporter 1'
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105135(CHEMBL542936 | N2-(3-((12-((3-((4Amino,6-(methylam...)
Affinity DataKi:  135nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089703(CHEMBL29507 | N-[4-(3-Nitrooxy-propyl)-phenyl]-[1,...)
Affinity DataKi:  200nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105123(CHEMBL544581 | N2-(3-((12-((3-((4Amino,6-(dimethyl...)
Affinity DataKi:  240nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105120(CHEMBL542932 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  410nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105124(CHEMBL553117 | N2-(3-[12-(3-[(4,6-Diamino-1,3,5-tr...)
Affinity DataKi:  500nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089708(2-(acetylamino)-N-{4-[(4,6-diamino-1,3,5-triazin-2...)
Affinity DataKi:  580nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105137(CHEMBL545281 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  600nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089698(2-(acetylamino)-N-[2-(6-amino-9H-purin-9-yl)ethyl]...)
Affinity DataKi:  620nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105121(CHEMBL542204 | N2-(3-((9-((3-((4-Amino-6-(methylam...)
Affinity DataKi:  750nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105125(CHEMBL541322 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  1.00E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089705(9-(2-Nitrooxy-ethyl)-9H-purin-6-ylamine | CHEMBL26...)
Affinity DataKi:  1.90E+3nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105139(CHEMBL544580 | N1,N9-Di(3-(((4,6-(dimethylamino-1,...)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105132(CHEMBL544335 | N2-(3-((12-((3-((4,6-Di(dimethylami...)
Affinity DataKi:  2.50E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105141(CHEMBL542698 | N2-(3-((12-((3-((4,6-Di(methylamino...)
Affinity DataKi:  3.20E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50366636(CHEMBL605462)
Affinity DataKi:  3.47E+3nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105133(CHEMBL541581 | N1,N9-Di(3-(((4-amino-6-(dimethylam...)
Affinity DataKi:  4.60E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105134(CHEMBL555240 | N1,N9-Di(3-(di((4,6-diamino-1,3,5-t...)
Affinity DataKi:  6.70E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105119(CHEMBL539797 | N2-(3-((9-((3-((4-Amino-6-(methylam...)
Affinity DataKi:  1.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM108256(CHEMBL2205239 | US8609833, 87)
Affinity DataKi:  1.23E+4nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105129(CHEMBL542208 | N2-(3-((9-((3-((4,6-Di(methylamino)...)
Affinity DataKi:  1.40E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105118(CHEMBL536324 | N1,N9-Di(3-(((4-amino-6-(dimethylam...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105142(CHEMBL554895 | N-{3-[9-(3-Amino-propylamino)-nonyl...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105138(CHEMBL543641 | N2-(3-[9-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  1.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50421414(CYMELARSEN | Cymelarsan)
Affinity DataKi:  2.29E+4nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105128(CHEMBL538778 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  2.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105143(CHEMBL544116 | N2-(3-((9-((3-((4,6-Di(dimethylamin...)
Affinity DataKi:  2.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105131(CHEMBL553511 | N1,N9-Di(3-(((4,6-(dimethylamino-1,...)
Affinity DataKi:  3.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105136(CHEMBL552613 | N2-(3-[2-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  5.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105130(CHEMBL543639 | N2-(3-[4-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  7.20E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105144(CHEMBL543884 | N1,N9-Di(3-(di((4,6-diamino-1,3,5-t...)
Affinity DataKi:  8.20E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089701(5,7-Diamino-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ol...)
Affinity DataKi:  1.17E+5nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105127(CHEMBL538771 | N2-(3-[4-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  1.25E+5nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105122(CHEMBL554860 | N2-(3-[2-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  1.63E+5nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089706(2-(acetylamino)-N-(6-aminopyridin-3-yl)-3-methyl-3...)
Affinity DataKi:  4.04E+5nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50366635(CHEMBL73188)
Affinity DataKi: >1.00E+6nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089704(CHEMBL25961 | nitrooxymethyl-benzene)
Affinity DataKi: >1.00E+6nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed