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Found 36 Enz. Inhib. hit(s) with Target = 'Adenylate kinase isoenzyme 1'
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367038(CHEMBL604815)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of AMP competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366480(ADENOSINE TRIPHOSPHATE | ATP)
Affinity DataKi:  5.70E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM18137(AMP | CHEMBL752 | US11185100, TABLE 7.3 | [(2R,3S,...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of AMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367104(CHEMBL607646)
Affinity DataKi:  6.00E+5nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367103(CHEMBL608483)
Affinity DataKi:  9.10E+5nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367098(CHEMBL607630)
Affinity DataKi:  1.40E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027451(CHEMBL3143591 | Phosphoric acid mono-[5-(6-amino-p...)
Affinity DataKi:  1.70E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367039(CHEMBL604398)
Affinity DataKi:  1.80E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367037(CHEMBL606008)
Affinity DataKi:  1.80E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367109(CHEMBL608484)
Affinity DataKi:  2.10E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367107(CHEMBL3244493 | CHEMBL610643)
Affinity DataKi:  2.30E+6nMAssay Description:Competitive Inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027448(CHEMBL3143581 | Phosphoric acid mono-[6-(6-amino-p...)
Affinity DataKi:  2.30E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367102(CHEMBL608353)
Affinity DataKi:  3.10E+6nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367099(CHEMBL606240 | CHEMBL609484)
Affinity DataKi:  3.20E+6nMAssay Description:Non-competitive Inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367110(CHEMBL609073)
Affinity DataKi:  3.70E+6nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367042(CHEMBL606221)
Affinity DataKi:  4.00E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027447(CHEMBL1229561 | Phosphoric acid mono-[5-(6-amino-p...)
Affinity DataKi:  4.10E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027446(CHEMBL3143582 | Phosphoric acid mono-[6-(6-amino-p...)
Affinity DataKi:  4.50E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367045(CHEMBL605010)
Affinity DataKi:  4.50E+6nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367046(CHEMBL604395)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATPnon competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367045(CHEMBL605010)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367108(CHEMBL1625734 | CHEMBL607918)
Affinity DataKi:  5.70E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010309(CHEMBL3251358)
Affinity DataKi:  6.10E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50027455(CHEMBL3143592 | Phosphoric acid mono-[6-(6-amino-p...)
Affinity DataKi:  6.50E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367100(CHEMBL607942)
Affinity DataKi:  1.10E+7nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367101(CHEMBL1788158)
Affinity DataKi:  1.50E+7nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367047(CHEMBL2368667)
Affinity DataKi:  1.50E+7nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367041(CHEMBL603556)
Affinity DataKi:  1.60E+7nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367041(CHEMBL603556)
Affinity DataKi:  1.60E+7nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  1.90E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II (AK-II) isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50222467(8-Bromo-Adenosine Mono Phosphate | CHEMBL1230617)
Affinity DataKi:  3.70E+7nMAssay Description:Non-competitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367105(CHEMBL608209)
Affinity DataKi:  5.20E+7nMAssay Description:Noncompetitive inhibitory constant of compound with Rat adenylate kinase M isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  8.20E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Oryctolagus cuniculus)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50277972(CHEMBL519503 | [5-(6-Amino-9-phenethyl-9H-purin-8-...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of rabbit muscle adenylate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Oryctolagus cuniculus)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50277565(5-(6-amino-9-neopentyl-9H-purin-8-yl)furan-2-ylpho...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of rabbit muscle adenylate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed