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Found 6 Enz. Inhib. hit(s) with Target = 'Aromatase [1-48]'
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  18nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85252(2,4-Trans-4'-hydroxy-4-imidazolyl-7-methoxyfla...)
Affinity DataIC50:  40nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85253(2,4-Trans-4',7-dihydroxy-4-imidazolyl-7-methox...)
Affinity DataIC50:  77nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85249(2,4-Trans-3'-hydroxy-4-imidazolyl-7-methoxyfla...)
Affinity DataIC50:  130nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85251(2,4-Trans-4'-cyano-4-imidazolyl-7-methoxyflava...)
Affinity DataIC50:  133nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85250(2,4-Trans-4'-chloro-4-imidazolyl-7-methoxyflav...)
Affinity DataIC50:  200nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed