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Found 125 Enz. Inhib. hit(s) with Target = 'Arylamine N-acetyltransferase'
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014986(CHEMBL3262086)
Affinity DataIC50:  120nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275074((Z)-5-(3',5'-Diiodo-4'-hydroxybenzylidene)-2-thiox...)
Affinity DataIC50:  138nMAssay Description:Inhibition of NAT1 in human ZR75 cell lysate assessed as acetylation of aryl amine using PABA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014986(CHEMBL3262086)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274859((Z)-3-Amino-5-(biphenyl-2'-ylmethylene)-2-thioxoth...)
Affinity DataIC50:  300nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275074((Z)-5-(3',5'-Diiodo-4'-hydroxybenzylidene)-2-thiox...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014944(CHEMBL3262085)
Affinity DataIC50:  430nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014944(CHEMBL3262085)
Affinity DataIC50:  540nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274853((Z)-5-(3'-Hydroxybenzylidene)-2-thioxothiazolidin-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014914(CHEMBL3262049)
Affinity DataIC50:  900nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275028((Z)-5-(4'-Methoxybenzylidene)-3-methyl-2-thioxothi...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014924(CHEMBL3262055)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50092273((Z)-5-(2'-Hydroxybenzylidene)-2-thioxothiazolidin-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274890((Z)-3-Amino-5-(4'-hydroxy-3',5-diiodobenzylidene)-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50368688(CHEMBL2047717)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Homo sapiens (human) arylamine N-acetyltransferase 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275069((Z)-5-Hexylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014931(CHEMBL3262062)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014912(CHEMBL1568345)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014914(CHEMBL3262049)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014922(CHEMBL3262053)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014912(CHEMBL1568345)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014924(CHEMBL3262055)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014913(CHEMBL3262048)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014943(CHEMBL3262084)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014943(CHEMBL3262084)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014938(CHEMBL3262077)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014922(CHEMBL3262053)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274887((Z)-5-(3',4'-Dichlorobenzylidene)-2-thioxothiazoli...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50240730((Z)-5-(4'-Hydroxy-3',5'-diiodobenzylidene)thiazoli...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014925(CHEMBL3262056)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274886((Z)-5-(2'-Methylbenzylidene)-2-thioxothiazolidin-4...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014913(CHEMBL3262048)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014942(CHEMBL3262082)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014930(CHEMBL3262061)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275064((Z)-3-Methyl-5-(2'-methylbenzylidene)-2-thioxothia...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274892((Z)-3-Methyl-5-(naphthalen-2'-ylmethylene)-2-thiox...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50181730((Z)-5-(4'-Chlorobenzylidene)-2-thioxothiazolidin-4...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275027((Z)-3-Amino-5-(2'-hydroxybenzylidene)-2-thioxothia...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014926(CHEMBL3262057)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014923(CHEMBL3262054)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274856((Z)-5-(4'-Biphenylmethylene)-3-methyl-2-thioxothia...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50181733((Z)-3-Amino-5-(4'-chlorobenzylidene)-2-thioxothiaz...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014942(CHEMBL3262082)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014987(CHEMBL3262087)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014938(CHEMBL3262077)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275066((Z)-5-(3'-Fluorobenzylidene)-2-thioxothiazolidin-4...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275070((Z)-5-Octylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014929(CHEMBL3262060)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275067((Z)-5-(3'-Fluorobenzylidene)-3-methyl-2-thioxothia...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274889((Z)-5-(4'-Hydroxy-3',5'-diiodobenzylidene)-3-methy...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human recombinant NAT1 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArylamine N-acetyltransferase 2(Mus musculus)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274898((Z)-5-Butylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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