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Found 5 Enz. Inhib. hit(s) with Target = 'Endothiapepsin'
TargetEndothiapepsin(Cryphonectria parasitica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50546276(CHEMBL4743297)
Affinity DataIC50:  54nMAssay Description:Inhibition of Endothia parasitica endothiapepsin using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothiapepsin(Cryphonectria parasitica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50546275(CHEMBL4797373)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of Endothia parasitica endothiapepsin using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEndothiapepsin(Cryphonectria parasitica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50546277(CHEMBL4747458)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of Endothia parasitica endothiapepsin using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothiapepsin(Cryphonectria parasitica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50514427(CHEMBL4452904)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of Cryphonectria parasitica Endothiapepsin using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 substrate by fluorescence screening assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothiapepsin(Cryphonectria parasitica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50226437(2-AMINO-6-(2-PHENYLETHYL)PYRIMIDIN-4(3H)-ONE | 2-a...)
Affinity DataKd:  2.20E+5nMAssay Description:Binding affinity to endothiapepsin by Biocore ISAMore data for this Ligand-Target Pair