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Found 3 Enz. Inhib. hit(s) with Target = 'Dimer of Gag-Pol polyprotein [600-1159,L699I,K702N,C879S]'
TargetDimer of Gag-Pol polyprotein [600-1159,L699I,K702N,C879S](Human immunodeficiency virus type 1)
Bar-Ilan University

LigandPNGBDBM16189(4-(3-Iodophenyl)-3-oxobutanenitrile | beta-ketonit...)
Affinity DataIC50:  9.40E+3nMpH: 7.5 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [600-1159,L699I,K702N,C879S](Human immunodeficiency virus type 1)
Bar-Ilan University

LigandPNGBDBM16196(4-(3-Bromo-4-chlorophenyl)-1H-imidazole-5-carboxam...)
Affinity DataIC50:  1.98E+4nMpH: 7.5 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [600-1159,L699I,K702N,C879S](Human immunodeficiency virus type 1)
Bar-Ilan University

LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  7.72E+4nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair