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Found 53 Enz. Inhib. hit(s) with Target = 'Xaa-Pro aminopeptidase 2'
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM197051(US9212206, III)
Affinity DataIC50:  3.70nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM197054(US9212206, VII)
Affinity DataIC50:  3.90nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM197053(US9212206, VI)
Affinity DataIC50:  9.70nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM197052(US9212206, V)
Affinity DataIC50:  26nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50:  130nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50:  230nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50:  230nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50:  310nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50:  430nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50:  560nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  660nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078398(2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolid...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078398(2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolid...)
Affinity DataIC50:  3.80E+3nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  4.10E+3nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078398(2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolid...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  9.20E+3nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078392((S)-1-((2R,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  1.90E+4nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078392((S)-1-((2R,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078392((S)-1-((2R,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  3.70E+4nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50351402(CHEMBL1819090)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  7.90E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  8.90E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  1.00E+5nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50:  1.50E+5nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50:  1.50E+5nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  3.90E+5nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50:  3.90E+5nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50:  3.90E+5nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50:  4.70E+5nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50:  6.00E+5nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50:  1.20E+6nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50:  1.70E+6nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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