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Found 47 Enz. Inhib. hit(s) with Target = 'Phosphopantetheine adenylyltransferase'
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82156(7-substituted pyrazoloquinolone, 15)
Affinity DataIC50:  5.00E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82152(7-substituted pyrazoloquinolone, 11)
Affinity DataIC50:  5.10E+3nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM50517256(CHEMBL4446301)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82151(7-substituted pyrazoloquinolone, 10)
Affinity DataIC50:  6.20E+3nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82157(7-substituted pyrazoloquinolone, 16)
Affinity DataIC50:  7.10E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50:  8.80E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82152(7-substituted pyrazoloquinolone, 11)
Affinity DataIC50:  1.10E+4nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50:  1.30E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82156(7-substituted pyrazoloquinolone, 15)
Affinity DataIC50:  1.40E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82160(6-substituted pyrazoloquinolone, 19)
Affinity DataIC50:  1.50E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82149(7-substituted pyrazoloquinolone, 8)
Affinity DataIC50:  1.70E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82154(7-substituted pyrazoloquinolone, 13)
Affinity DataIC50:  2.00E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82151(7-substituted pyrazoloquinolone, 10)
Affinity DataIC50:  2.20E+4nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82157(7-substituted pyrazoloquinolone, 16)
Affinity DataIC50:  4.90E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82164(6-substituted pyrazoloquinolone, 23)
Affinity DataIC50:  4.90E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82161(6-substituted pyrazoloquinolone, 20)
Affinity DataIC50:  5.40E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50: >6.50E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82149(7-substituted pyrazoloquinolone, 8)
Affinity DataIC50: >7.50E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82155(7-substituted pyrazoloquinolone, 14)
Affinity DataIC50:  9.20E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82164(6-substituted pyrazoloquinolone, 23)
Affinity DataIC50:  9.30E+4nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82162(6-substituted pyrazoloquinolone, 21)
Affinity DataIC50:  1.00E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM50517254(CHEMBL4553617)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM50517257(CHEMBL4584904)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82150(7-substituted pyrazoloquinolone, 9)
Affinity DataIC50:  1.03E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82165(3-substituted pyrazoloquinolone, 24)
Affinity DataIC50:  1.06E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82162(6-substituted pyrazoloquinolone, 21)
Affinity DataIC50:  1.21E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82163(6-substituted pyrazoloquinolone, 22)
Affinity DataIC50:  1.24E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82163(6-substituted pyrazoloquinolone, 22)
Affinity DataIC50: >1.25E+5nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82152(7-substituted pyrazoloquinolone, 11)
Affinity DataIC50: >1.37E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82158(7-substituted pyrazoloquinolone, 17)
Affinity DataIC50: >1.50E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82157(7-substituted pyrazoloquinolone, 16)
Affinity DataIC50:  1.57E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82159(4-substituted pyrazoloquinolone, 18)
Affinity DataIC50:  1.60E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82154(7-substituted pyrazoloquinolone, 13)
Affinity DataIC50:  1.66E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82163(6-substituted pyrazoloquinolone, 22)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82161(6-substituted pyrazoloquinolone, 20)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82160(6-substituted pyrazoloquinolone, 19)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82165(3-substituted pyrazoloquinolone, 24)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82158(7-substituted pyrazoloquinolone, 17)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82150(7-substituted pyrazoloquinolone, 9)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82147(7-substituted pyrazoloquinolone, 6)
Affinity DataIC50: >1.67E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82161(6-substituted pyrazoloquinolone, 20)
Affinity DataIC50:  2.00E+5nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82151(7-substituted pyrazoloquinolone, 10)
Affinity DataIC50:  2.09E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82164(6-substituted pyrazoloquinolone, 23)
Affinity DataIC50:  2.12E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82147(7-substituted pyrazoloquinolone, 6)
Affinity DataIC50: >2.30E+5nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82148(7-substituted pyrazoloquinolone, 7)
Affinity DataIC50:  2.44E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82156(7-substituted pyrazoloquinolone, 15)
Affinity DataIC50:  2.49E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82147(7-substituted pyrazoloquinolone, 6)
Affinity DataIC50:  2.53E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed