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Found 68 Enz. Inhib. hit(s) with Target = 'Protein kinase domain-containing protein'
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265061(4-(6-((trans)-4-hydroxycyclohexylamino)imidazo[1,2...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265061(4-(6-((trans)-4-hydroxycyclohexylamino)imidazo[1,2...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265063(4-(6-((+/-)-2-hydroxycyclohexylamino)imidazo[1,2-b...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265063(4-(6-((+/-)-2-hydroxycyclohexylamino)imidazo[1,2-b...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265062(4-(6-((+/-)-3-hydroxycyclohexylamino)imidazo[1,2-b...)
Affinity DataIC50:  260nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265062(4-(6-((+/-)-3-hydroxycyclohexylamino)imidazo[1,2-b...)
Affinity DataIC50:  260nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264942((S)-4-(6-(1-hydroxy-3-methylbutan-2-ylamino)imidaz...)
Affinity DataIC50:  280nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264942((S)-4-(6-(1-hydroxy-3-methylbutan-2-ylamino)imidaz...)
Affinity DataIC50:  280nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265064(4-(6-(cyclohexylamino)imidazo[1,2-b]pyridazin-3-yl...)
Affinity DataIC50:  340nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265064(4-(6-(cyclohexylamino)imidazo[1,2-b]pyridazin-3-yl...)
Affinity DataIC50:  340nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265025((S)-4-(6-(1-hydroxypropan-2-ylamino)imidazo[1,2-b]...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265025((S)-4-(6-(1-hydroxypropan-2-ylamino)imidazo[1,2-b]...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264906(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  579nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264906(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  580nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264905(4-(6-((tetrahydrofuran-2-yl)methylamino)imidazo[1,...)
Affinity DataIC50:  750nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264905(4-(6-((tetrahydrofuran-2-yl)methylamino)imidazo[1,...)
Affinity DataIC50:  750nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264943((S)-4-(6-(1-hydroxy-3-methylbutan-2-ylamino)imidaz...)
Affinity DataIC50:  769nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264943((S)-4-(6-(1-hydroxy-3-methylbutan-2-ylamino)imidaz...)
Affinity DataIC50:  770nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264902(4-(6-(pyridin-3-ylmethylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  809nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264902(4-(6-(pyridin-3-ylmethylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  810nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265060((S)-4-(6-(1-methoxypropan-2-ylamino)imidazo[1,2-b]...)
Affinity DataIC50:  820nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265060((S)-4-(6-(1-methoxypropan-2-ylamino)imidazo[1,2-b]...)
Affinity DataIC50:  820nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265026((R)-4-(6-(1-hydroxypropan-2-ylamino)imidazo[1,2-b]...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265027(4-(6-(2-hydroxyethylamino)imidazo[1,2-b]pyridazin-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265027(4-(6-(2-hydroxyethylamino)imidazo[1,2-b]pyridazin-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265026((R)-4-(6-(1-hydroxypropan-2-ylamino)imidazo[1,2-b]...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50486604(CHEMBL2235667)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264904(4-(6-((4-fluorobenzyl)(methyl)amino)imidazo[1,2-b]...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50486603(CHEMBL2235668)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264983(4-(6-((4-fluorobenzyl)(methyl)amino)imidazo[1,2-b]...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264903(4-(6-(methyl(pyridin-3-ylmethyl)amino)imidazo[1,2-...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264903(4-(6-(methyl(pyridin-3-ylmethyl)amino)imidazo[1,2-...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265059(4-(6-(2-methoxyethylamino)imidazo[1,2-b]pyridazin-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265059(4-(6-(2-methoxyethylamino)imidazo[1,2-b]pyridazin-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50486598(CHEMBL2236083)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265101((+/-)-4-(6-(piperidin-3-ylamino)imidazo[1,2-b]pyri...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265104((R)-1-(3-morpholinophenyl)ethanamine | CHEMBL49756...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265104((R)-1-(3-morpholinophenyl)ethanamine | CHEMBL49756...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264944((S)-2-(3-(4-(hydroxymethyl)phenyl)imidazo[1,2-b]py...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264944((S)-2-(3-(4-(hydroxymethyl)phenyl)imidazo[1,2-b]py...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264870(CHEMBL524106 | N-(pyridin-3-ylmethyl)-3-(pyridin-4...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264870(CHEMBL524106 | N-(pyridin-3-ylmethyl)-3-(pyridin-4...)
Affinity DataIC50:  7.91E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265102(4-(6-(4-morpholinobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265102(4-(6-(4-morpholinobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264869(3-(4-methoxyphenyl)-N-(pyridin-3-ylmethyl)imidazo[...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264869(3-(4-methoxyphenyl)-N-(pyridin-3-ylmethyl)imidazo[...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50486602(CHEMBL2235669)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Plasmodium falciparum protein kinase 7More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264984((4-(6-((4-fluorobenzyl)(methyl)amino)imidazo[1,2-b...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50264945((S)-2-(4-(6-(1-hydroxy-3-methylbutan-2-ylamino)imi...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase domain-containing protein(Plasmodium falciparum)TBA
LigandPNGBDBM50265105((S)-1-(3-morpholinophenyl)ethanamine | CHEMBL44675...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum PK7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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