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Found 123 Enz. Inhib. hit(s) with Target = 'Phospholipase A2 group V'
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601469(CHEMBL5172164)
Affinity DataIC50:  10nMAssay Description:Inhibition of human group V phospholipase A2 expressed in Escherichia coli BL21(DE3) cells incubated for 10 to 20 mins cells by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50601469(CHEMBL5172164)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse group V phospholipase A2 incubated for 10 to 20 mins cells by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263002((2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-6,7-benz...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50263002((2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-6,7-benz...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055391(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-ind...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055391(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-ind...)
Affinity DataIC50:  57nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50262842(Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzy...)
Affinity DataIC50:  60nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263000(2-(1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)-N-(...)
Affinity DataIC50:  70nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50262842(Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50274336(1-{3-Dodecanoyl-2,4,6-trihydroxy-5-[7-hydroxy-2-(4...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  124nMAssay Description:Inhibition of recombinant human sPLA2-5 expressed in Escherichia coli BL21(DE3) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50263000(2-(1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)-N-(...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  170nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50458608(CHEMBL4205008)
Affinity DataIC50:  180nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50458608(CHEMBL4205008)
Affinity DataIC50:  180nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50333788((S)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50186585(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-6-meth...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50458612(CHEMBL4214052)
Affinity DataIC50:  510nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50458606(CHEMBL4205511)
Affinity DataIC50:  510nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274336(1-{3-Dodecanoyl-2,4,6-trihydroxy-5-[7-hydroxy-2-(4...)
Affinity DataIC50:  520nMAssay Description:Inhibition of mouse sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50274337(1-(3-Dodecanoyl-2,4,6-trihydroxy-5-methyl-phenyl)-...)
Affinity DataIC50:  530nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  620nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  660nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50458609(CHEMBL4213094)
Affinity DataIC50:  720nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50186585(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-6-meth...)
Affinity DataIC50:  750nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055383((3-Aminooxalyl-1-benzyl-2-methyl-1H-indol-4-yloxy)...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50186586(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2,6-dimethyl-1...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50186586(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2,6-dimethyl-1...)
Affinity DataIC50:  850nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055383((3-Aminooxalyl-1-benzyl-2-methyl-1H-indol-4-yloxy)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50591714(CHEMBL5200953)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of human PLA2G5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50149981(CHEMBL3769794)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human group 5 secreted phospholipase A2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50591712(CHEMBL5194852)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of human PLA2G5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50333789((R)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50591713(CHEMBL5207115)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of human PLA2G5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50263053(2-(3-Biphenyl-2-ylmethyl-2-ethyl-8-methoxy-indoliz...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274388(2-Phenyl-1-(2,4,6-trihydroxy-3-methyl-5-phenylacet...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of mouse sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274389(1-(3-acetyl-2,4,6-trihydroxy-5-methylphenyl)dodeca...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of mouse sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50274387(1-(3-Acetyl-2,4,6-trihydroxy-5-methyl-phenyl)-etha...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50274388(2-Phenyl-1-(2,4,6-trihydroxy-3-methyl-5-phenylacet...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50274389(1-(3-acetyl-2,4,6-trihydroxy-5-methylphenyl)dodeca...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Mus musculus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274441(1-(3-Acetyl-5-dodecyl-2,4,6-trihydroxy-phenyl)-eth...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of mouse sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50274441(1-(3-Acetyl-5-dodecyl-2,4,6-trihydroxy-phenyl)-eth...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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