TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 22.7nMAssay Description:Inhibition of human MAK using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 28.7nMAssay Description:Inhibition of human MAK using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAK using RRRFRPASPLRGP as substrate after 120 mins in presence of [gamma-33ATP] by radiometric scintillation countin...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.30E+3nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 890nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 97nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MAK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MAK kinase domainMore data for this Ligand-Target Pair