Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with Target = 'Type 1 fimbiral adhesin FimH'
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197181(CHEMBL3899291)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197180(CHEMBL3945119)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197182(CHEMBL3961517)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197178(CHEMBL3894223)
Affinity DataIC50:  80nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197172(CHEMBL3936194)
Affinity DataIC50:  130nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197173(CHEMBL3923903)
Affinity DataIC50:  140nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197185(CHEMBL2058201)
Affinity DataIC50:  150nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197174(CHEMBL3908258)
Affinity DataIC50:  250nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197176(CHEMBL3892524)
Affinity DataIC50:  340nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197183(CHEMBL3973443)
Affinity DataIC50:  600nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197175(CHEMBL3927866)
Affinity DataIC50:  900nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197179(CHEMBL1172856)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347464(CHEMBL1802187)
Affinity DataIC50:  9.00E+3nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347465(CHEMBL1802185)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197177(CHEMBL3953852)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347452(CHEMBL1802190)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347457(CHEMBL1802189)
Affinity DataIC50:  1.70E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347450(CHEMBL1802194)
Affinity DataIC50:  3.10E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347454(CHEMBL1171678)
Affinity DataIC50:  3.30E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50197184(CHEMBL3955472)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of Escherichia coli UTI89 FimH-mediated biofilm formation after 48 hrs by crystal violet staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347455(CHEMBL1802188)
Affinity DataIC50:  4.10E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347449(CHEMBL1171278)
Affinity DataIC50:  4.20E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347453(CHEMBL1802186)
Affinity DataIC50:  4.50E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347459(CHEMBL1802193)
Affinity DataIC50:  4.50E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
Fimbrion Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataIC50:  7.71E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed