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Found 57 Enz. Inhib. hit(s) with Target = 'Voltage-dependent calcium channel alpha-2 delta subunit'
LigandPNGBDBM50305900((+)-2-((1S,5S,6R)-6-(aminomethyl)bicyclo[3.2.0]hep...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305887(3,4-trans-2-(1-(aminomethyl)-3,4-dimethylcyclopent...)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305894((+/-)-2-((6S)-6-(aminomethyl)bicyclo[3.2.0]heptan-...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304703(2-((3R)-1-(aminomethyl)-3-propylcyclopentyl)acetic...)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304707(2-((1R,3R)-1-(aminomethyl)-3-methylcyclopentyl)ace...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305885(CHEMBL595172 | cis-2-((1R,5S)-3-(aminomethyl)bicyc...)
Affinity DataIC50:  38nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305899((-)-2-((1R,5R,6S)-6-(aminomethyl)bicyclo[3.2.0]hep...)
Affinity DataIC50:  46nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304702(2-((3R)-1-(aminomethyl)-3-ethylcyclopentyl)acetic ...)
Affinity DataIC50:  53nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304693(2-(1-(aminomethyl)-3-ethylcyclopentyl)acetic acid ...)
Affinity DataIC50:  55nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304694(2-(1-(aminomethyl)-3-propylcyclopentyl)acetic acid...)
Affinity DataIC50:  69nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080153((1-Aminomethyl-cyclohexyl)-acetic acid | 2-(1-(ami...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]gabapentin from alpha-2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
LigandPNGBDBM50304708(2-((1S,3R)-1-(aminomethyl)-3-methylcyclopentyl)ace...)
Affinity DataIC50:  71nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50164279((S)-3-(aminomethyl)-5-methylhexanoic acid | (S)-3-...)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50164279((S)-3-(aminomethyl)-5-methylhexanoic acid | (S)-3-...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304692(2-(1-(aminomethyl)-3-methylcyclopentyl)acetic acid...)
Affinity DataIC50:  82nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304701(2-((3R)-1-(aminomethyl)-3-methylcyclopentyl)acetic...)
Affinity DataIC50:  88nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50168499((1-((1H-tetrazol-5-yl)methyl)cycloheptyl)methanami...)
Affinity DataIC50:  100nMAssay Description:Displacement of [3H]gabapentin from alpha-2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305886(2-((3R,4S)-1-(aminomethyl)-3,4-dimethylcyclopentyl...)
Affinity DataIC50:  107nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212317((1-((1H-tetrazol-5-yl)methyl)cyclohexyl)methanamin...)
Affinity DataIC50:  108nMAssay Description:Displacement of [3H]gabapentin from alpha-2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080153((1-Aminomethyl-cyclohexyl)-acetic acid | 2-(1-(ami...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
LigandPNGBDBM50171790((S)-3-(aminomethyl)-4-(furan-2-yl)butanoic acid | ...)
Affinity DataIC50:  178nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305884(CHEMBL609569 | cis-2-((1R,5S)-3-(aminomethyl)bicyc...)
Affinity DataIC50:  332nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304691(CHEMBL610734 | Gababutin)
Affinity DataIC50:  420nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171795(3-(aminomethyl)-4-(furan-2-yl)butanoic acid | CHEM...)
Affinity DataIC50:  421nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171794(3-(aminomethyl)-4-(furan-3-yl)butanoic acid | CHEM...)
Affinity DataIC50:  518nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305897((+/-)-2-((7S)-7-(aminomethyl)bicyclo[4.2.0]octan-7...)
Affinity DataIC50:  600nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304695(2-(1-(aminomethyl)-3-butylcyclopentyl)acetic acid ...)
Affinity DataIC50:  690nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304705(2-((3S)-1-(aminomethyl)-3-ethylcyclopentyl)acetic ...)
Affinity DataIC50:  706nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305892(2-((2R,3aR)-2-(aminomethyl)octahydro-1H-inden-2-yl...)
Affinity DataIC50:  720nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304696(2-(1-(aminomethyl)-3-isobutylcyclopentyl)acetic ac...)
Affinity DataIC50:  760nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171796(3-(aminomethyl)-4-(thiophen-3-yl)butanoic acid | C...)
Affinity DataIC50:  832nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304706(2-((3S)-1-(aminomethyl)-3-propylcyclopentyl)acetic...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304704(2-((3S)-1-(aminomethyl)-3-methylcyclopentyl)acetic...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171792((R)-3-(aminomethyl)-4-(furan-2-yl)butanoic acid | ...)
Affinity DataIC50:  1.46E+3nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50168498((S)-2-((1H-tetrazol-5-yl)methyl)-4-methylpentan-1-...)
Affinity DataIC50:  1.59E+3nMAssay Description:Displacement of [3H]gabapentin from alpha-2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171789(3-(aminomethyl)-4-(thiophen-2-yl)butanoic acid | C...)
Affinity DataIC50:  2.14E+3nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50168502((1-((1H-tetrazol-5-yl)methyl)cyclooctyl)methanamin...)
Affinity DataIC50:  2.36E+3nMAssay Description:Displacement of [3H]gabapentin from alpha-2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305890(2-((2R,3aR)-2-(aminomethyl)octahydropentalen-2-yl)...)
Affinity DataIC50:  2.60E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305895((+/-)-2-((6R)-6-(aminomethyl)bicyclo[3.2.0]heptan-...)
Affinity DataIC50:  2.80E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305884(CHEMBL609569 | cis-2-((1R,5S)-3-(aminomethyl)bicyc...)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305898((+/-)-2-((7R)-7-(aminomethyl)bicyclo[4.2.0]octan-7...)
Affinity DataIC50:  3.09E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304690(2-(1-(aminomethyl)-3,3-dimethylcyclopentyl)acetic ...)
Affinity DataIC50:  3.18E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304698(2-(1-(aminomethyl)-3-phenylcyclopentyl)acetic acid...)
Affinity DataIC50:  5.06E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304700(2-(1-(aminomethyl)-3-phenethylcyclopentyl)acetic a...)
Affinity DataIC50:  6.23E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305896((+/-)-2-((1S)-1-(aminomethyl)octahydropentalen-1-y...)
Affinity DataIC50:  7.18E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304699(2-(1-(aminomethyl)-3-benzylcyclopentyl)acetic acid...)
Affinity DataIC50:  9.28E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305893(2-((2S,3aR)-2-(aminomethyl)octahydro-1H-inden-2-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305889((+/-)-2-(2-(aminomethyl)octahydro-1H-inden-2-yl)ac...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305888((+/-)-2-(2-(aminomethyl)octahydropentalen-2-yl)ace...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304697(2-(1-(aminomethyl)-3-tert-butylcyclopentyl)acetic ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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