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Found 82 Enz. Inhib. hit(s) with Target = 'Transmembrane protease serine 11D'
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420334(CHEMBL2086421)
Affinity DataKi:  8.40nMAssay Description:Tight binding inhibition of human TMPRSS11D expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 15 mins prior ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349355(CHEMBL1809213)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349344(CHEMBL1809250)
Affinity DataKi:  14nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349345(CHEMBL1809251)
Affinity DataKi:  15nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349333(CHEMBL1809238)
Affinity DataKi:  17nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50324475(Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzy...)
Affinity DataKi:  19nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349346(CHEMBL1809252)
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349347(CHEMBL1809253)
Affinity DataKi:  23nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349348(CHEMBL1809254)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349349(CHEMBL1809255)
Affinity DataKi:  34nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349350(CHEMBL1809256)
Affinity DataKi:  34nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349357(CHEMBL1809214)
Affinity DataKi:  36nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349334(CHEMBL1809239)
Affinity DataKi:  38nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349361(CHEMBL1809215)
Affinity DataKi:  38nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349358(CHEMBL1809216)
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349335(CHEMBL1809240)
Affinity DataKi:  43nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349351(CHEMBL1809257)
Affinity DataKi:  47nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349360(CHEMBL1809212)
Affinity DataKi:  51nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349362(CHEMBL1809217)
Affinity DataKi:  53nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50323871((6S,9S,12S,15S)-1,20-diamino-12-(3-amino-3-oxoprop...)
Affinity DataKi:  54.3nMAssay Description:Inhibition of human HAT by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349352(CHEMBL1809258)
Affinity DataKi:  57nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349363(CHEMBL1809218)
Affinity DataKi:  63nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349336(CHEMBL1809241)
Affinity DataKi:  68nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349337(CHEMBL1809242)
Affinity DataKi:  73nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349364(CHEMBL1809219)
Affinity DataKi:  76nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50231520((R)-N-[(S)-1-(4-carbamimidoyl-benzylcarbamoyl)-2-h...)
Affinity DataKi:  78nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349365(CHEMBL1809220)
Affinity DataKi:  98nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50324477(Benzylsulfonyl-D-cyclohexylalanyl-proline-(4-amidi...)
Affinity DataKi:  108nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50323872((6S,9S,12S,15S)-1,19-diamino-9-(3-amino-3-oxopropy...)
Affinity DataKi:  112nMAssay Description:Inhibition of human HAT by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349367(CHEMBL1809234)
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349371(CHEMBL1809243)
Affinity DataKi:  135nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349338(CHEMBL1809244)
Affinity DataKi:  149nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349339(CHEMBL1809245)
Affinity DataKi:  158nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349368(CHEMBL1809235)
Affinity DataKi:  168nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349340(CHEMBL1809246)
Affinity DataKi:  183nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349341(CHEMBL1809247)
Affinity DataKi:  202nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349342(CHEMBL1809248)
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349343(CHEMBL1809249)
Affinity DataKi:  221nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349369(CHEMBL1809236)
Affinity DataKi:  311nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349353(CHEMBL1809259)
Affinity DataKi:  422nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349359(CHEMBL1809211)
Affinity DataKi:  430nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349372(CHEMBL1809260)
Affinity DataKi:  457nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349354(CHEMBL1809261)
Affinity DataKi:  512nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50349370(CHEMBL1809237)
Affinity DataKi:  1.43E+3nMAssay Description:Inhibition of human recombinant airway trypsin-like protease HAT using D-cyclohexylalanine-Pro-Arg-AMC as substrate by fluorescence plate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM441788(US10640533, Identification number CX13-606 | US106...)
Affinity DataIC50:  186nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM441788(US10640533, Identification number CX13-606 | US106...)
Affinity DataIC50:  297nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM441779(US10640533, Identification number CX13-133 | US106...)
Affinity DataIC50:  443nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM441779(US10640533, Identification number CX13-133 | US106...)
Affinity DataIC50:  455nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM441789(US10640533, Identification number CX13-608 | US106...)
Affinity DataIC50:  490nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM441789(US10640533, Identification number CX13-608 | US106...)
Affinity DataIC50:  542nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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