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Found 3 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase Su(var)3-9'
TargetHistone-lysine N-methyltransferase Su(var)3-9(Drosophila melanogaster)
TBA

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant Drosophila melanogaster SUV39 by radioactive filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase Su(var)3-9(Drosophila melanogaster)
TBA

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  600nMAssay Description:Inhibition of Drosophila melanogaster SU(VAR)3-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase Su(var)3-9(Drosophila melanogaster)
TBA

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  600nMAssay Description:Inhibition of Drosophila melanogaster Histone-lysine N-methyltransferase Su(var)3-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed