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Found 45 Enz. Inhib. hit(s) with Target = 'IgA-specific serine endopeptidase autotransporter'
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016709(2-({1-[1-(2-Acetylamino-3-hydroxy-butyryl)-pyrroli...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016729(1-[1-(2-Acetylamino-3-hydroxy-butyryl)-pyrrolidine...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016716(Acetylprolylprolylthreonylprolinamide(AcPPTPNH2) |...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016727(1-(2-{[1-(1-Acetyl-pyrrolidine-2-carbonyl)-pyrroli...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016712(1-{3-Hydroxy-2-[(pyrrolidine-2-carbonyl)-amino]-bu...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016710(1-{1-[2-(2-Acetylamino-3-hydroxy-propionylamino)-3...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016724(2-[(1-{2-[(1-Acetyl-pyrrolidine-2-carbonyl)-amino]...)
Affinity DataIC50:  2.38E+4nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016714(1-(3-Hydroxy-2-{[1-(pyrrolidine-2-carbonyl)-pyrrol...)
Affinity DataIC50:  4.05E+4nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016717(1-{1-[2-(2-Amino-3-hydroxy-propionylamino)-3-hydro...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367755(CHEMBL2369567)
Affinity DataIC50:  1.70E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinase assayed in 40% TFEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016719(1-(2-{[1-(2-Acetylamino-3-hydroxy-butyryl)-pyrroli...)
Affinity DataIC50:  1.83E+5nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367751(CHEMBL2369563)
Affinity DataIC50:  2.00E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367755(CHEMBL2369567)
Affinity DataIC50:  2.00E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinase in 40% TFEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367751(CHEMBL2369563)
Affinity DataIC50:  2.00E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367754(CHEMBL2369558)
Affinity DataIC50:  2.60E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367754(CHEMBL2369558)
Affinity DataIC50:  2.60E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367756(CHEMBL2369562)
Affinity DataIC50:  3.10E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367758(CHEMBL2369564)
Affinity DataIC50:  3.10E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367756(CHEMBL2369562)
Affinity DataIC50:  3.10E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367753(CHEMBL2369569)
Affinity DataIC50:  4.00E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367753(CHEMBL2369569)
Affinity DataIC50:  4.00E+5nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016711(1-[1-(2-Amino-3-hydroxy-butyryl)-pyrrolidine-2-car...)
Affinity DataIC50:  4.19E+5nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016725(2-[(1-{2-[(1-Acetyl-pyrrolidine-2-carbonyl)-amino]...)
Affinity DataIC50:  6.75E+5nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016720(3-Hydroxy-2-[(1-{3-hydroxy-2-[(pyrrolidine-2-carbo...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016721(Acetylprolylthreonylprolylserinamide(AcPTPSNH2) | ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016732(Acetylthreonylprolylserylprolinamide(AcTPSPNH2) | ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016730(2-({1-[1-(2-Amino-3-hydroxy-butyryl)-pyrrolidine-2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016722(1-{1-[2-(2-Amino-3-hydroxy-propionylamino)-3-hydro...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016728(CHEMBL420584 | Prolylprolylthreonylprolinamide(PPT...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016723(CHEMBL310908 | Threonylprolylserylprolinamide(TPSP...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016726(1-{1-[2-(2-Acetylamino-3-hydroxy-propionylamino)-3...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016715(Acetylprolylserylprolylserinamide(AcPSPSNH2) | CHE...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016713(3-Hydroxy-2-[(1-{3-hydroxy-2-[(pyrrolidine-2-carbo...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016718(1-{3-Hydroxy-2-[(pyrrolidine-2-carbonyl)-amino]-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367750(CHEMBL2369561)
Affinity DataIC50:  1.03E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367750(CHEMBL2369561)
Affinity DataIC50:  1.03E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367757(CHEMBL2369560)
Affinity DataIC50:  1.57E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367757(CHEMBL2369560)
Affinity DataIC50:  1.57E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367749(CHEMBL2369559)
Affinity DataIC50:  1.81E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367749(CHEMBL2369559)
Affinity DataIC50:  1.81E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367759(CHEMBL2369557)
Affinity DataIC50:  3.30E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367752(CHEMBL3037869)
Affinity DataIC50:  5.15E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367748(CHEMBL2369568)
Affinity DataIC50:  9.35E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50367748(CHEMBL2369568)
Affinity DataIC50:  9.35E+6nMAssay Description:Tested for inhibitory activity against IgA1 proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIgA-specific serine endopeptidase autotransporter(Neisseria gonorrhoeae)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50016731(1-(2-{[1-(2-Amino-3-hydroxy-butyryl)-pyrrolidine-2...)
Affinity DataIC50:  3.31E+7nMAssay Description:Inhibitory concentration against type 1 IgA1 proteinases secreted by Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed