Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with Target = 'Integrin beta-3'
TargetIntegrin beta-3(Mus musculus)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50083811(3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at mouse endothelial alpha2bbeta3 integrin receptor by cell adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50004058((2S)-2-(butylsulfonylamino)-3-[4-(4-piperidin-4-yl...)
Affinity DataIC50:  130nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50004058((2S)-2-(butylsulfonylamino)-3-[4-(4-piperidin-4-yl...)
Affinity DataIC50:  136nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50568659(CHEMBL4861415)
Affinity DataIC50:  603nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50568659(CHEMBL4861415)
Affinity DataIC50:  610nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50568658(CHEMBL4853717)
Affinity DataIC50:  890nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50568658(CHEMBL4853717)
Affinity DataIC50:  897nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin beta-3/subunit alpha 2b(Rattus norvegicus)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50453875(CHEMBL1811964)
Affinity DataEC50:  1.66E+3nMAssay Description:Binding affinity to GP2b/3a in rat blood assessed as conformational change by measuring soluble GP2b/3a levels after 12 hrs by UV-spectrophotometric ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin beta-3(Rattus norvegicus)
University Of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453876(CHEMBL4212580)
Affinity DataEC50:  1.16E+3nMAssay Description:Binding affinity to GP2b/3a in rat blood assessed as conformational change by measuring soluble GP2b/3a levels after 12 hrs by UV-spectrophotometric ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed