Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Probable JmjC domain-containing histone demethylation protein 2C'
TargetProbable JmjC domain-containing histone demethylation protein 2C(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of KDM3C (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable JmjC domain-containing histone demethylation protein 2C(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594964(CHEMBL5193187)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to CM7 sensor chip immobilized partial-length JMJD1C (2274 to 2498 residues) (unknown origin) expressed in Escherichia coli assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable JmjC domain-containing histone demethylation protein 2C(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594965(CHEMBL5173150)
Affinity DataKd:  8.06E+3nMAssay Description:Binding affinity to CM7 sensor chip immobilized partial-length JMJD1C (2274 to 2498 residues) (unknown origin) expressed in Escherichia coli assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable JmjC domain-containing histone demethylation protein 2C(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594963(CHEMBL5191875)
Affinity DataKd:  2.67E+4nMAssay Description:Binding affinity to CM7 sensor chip immobilized partial-length JMJD1C (2274 to 2498 residues) (unknown origin) expressed in Escherichia coli assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed