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Found 155 Enz. Inhib. hit(s) with Target = 'Pancreatic alpha-amylase'
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM223314(YPYSCWARHVRIREN | piHA-D1)
Affinity DataKi:  1nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM223315(YPYSCWVRHSDPHKF | piHA-D3)
Affinity DataKi:  2.70nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM223316(YPYSCWVRH | piHA-Dm)
Affinity DataKi:  7nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120854(CHEMBL3618493)
Affinity DataKi:  8nMAssay Description:Competitive inhibition of human pancreatic alpha-amylase by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163646(Montbretin A (MbA))
Affinity DataKi:  8.10nM ΔG°:  -47.0kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163647(MbA-G (1))
Affinity DataKi:  9.10nM ΔG°:  -46.7kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120850(CHEMBL3618491)
Affinity DataKi:  12nMAssay Description:Inhibition of human pancreatic alpha-amylaseMore data for this Ligand-Target Pair
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120851(CHEMBL1233515)
Affinity DataKi:  12nMAssay Description:Inhibition of human pancreatic alpha-amylaseMore data for this Ligand-Target Pair
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120843(CHEMBL3616594)
Affinity DataKi:  14nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120842(CHEMBL3618489)
Affinity DataKi:  15nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163648(MbA-R (2))
Affinity DataKi:  21.3nM ΔG°:  -44.5kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120844(CHEMBL3616595)
Affinity DataKi:  42nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163649(MbA-RX (3))
Affinity DataKi:  42.4nM ΔG°:  -42.8kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120852(CHEMBL1230193)
Affinity DataKi:  75nMAssay Description:Inhibition of human pancreatic alpha-amylaseMore data for this Ligand-Target Pair
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163650(MbA-GR (4))
Affinity DataKi:  79.3nM ΔG°:  -41.2kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163651(MbA-GRX (5) | mini-MbA)
Affinity DataKi:  93.3nM ΔG°:  -40.8kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163652(MbA-C (6))
Affinity DataKi:  730nM ΔG°:  -35.6kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120848(CHEMBL3618488)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163653(MbA-CG (7))
Affinity DataKi:  2.24E+3nM ΔG°:  -32.8kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120855(CHEMBL3618494)
Affinity DataKi:  3.60E+3nMAssay Description:Competitive inhibition of human pancreatic alpha-amylase by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120856(CHEMBL3618495)
Affinity DataKi:  6.10E+3nMAssay Description:Competitive inhibition of human pancreatic alpha-amylase by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50499987(CHEMBL3742315)
Affinity DataKi:  1.17E+4nMAssay Description:Non-competitive inhibition of porcine pancreatic alpha-amylase by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163656(3-O-(6-(4-(Caffeamidomethyl)-triazolyl)hexyl)querc...)
Affinity DataKi:  1.39E+4nM ΔG°:  -28.2kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120839(CHEMBL1234040)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human pancreatic alpha-amylase assessed as hydrolysis of G3F by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM92367(GPESB15)
Affinity DataKi:  3.36E+4nM ΔG°:  -26.6kJ/mole IC50:  3.58E+4nMpH: 7.0 T: 2°CAssay Description:To test whether GCTs share a common binding pocket on PPA with acarbose, we performed an experiment according to the method of Yonetani and Theorell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50451094(Ascorbyl Palmitate | Ascorbyl palmitate (E5) | E30...)
Affinity DataKi: <4.00E+4nMAssay Description:Inhibitory constant against Alpha-amylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50090254((R)-5-((S)-2,2-Dimethyl-[1,3]dioxolan-4-yl)-3,4-di...)
Affinity DataKi: <4.00E+4nMAssay Description:Inhibitory constant against Alpha-amylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50351096(ASCORBIC ACID)
Affinity DataKi:  4.34E+4nMAssay Description:Inhibitory constant against Alpha-amylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163654(MbA-CR (8))
Affinity DataKi:  4.68E+4nM ΔG°:  -25.1kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM29143(CHEMBL7976 | Chalcone 1 | Chalcone, 13 | cid_63776...)
Affinity DataKi:  4.80E+4nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using soluble starch as substrate after 30 mins by Bernfeld methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM163655(MbA-CGR (9))
Affinity DataKi:  1.28E+5nM ΔG°:  -22.6kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM92366(GPESB14)
Affinity DataKi:  2.04E+5nM ΔG°:  -21.9kJ/mole IC50:  8.89E+4nMpH: 7.0 T: 2°CAssay Description:To test whether GCTs share a common binding pocket on PPA with acarbose, we performed an experiment according to the method of Yonetani and Theorell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM92365(GPESB11)
Affinity DataKi:  2.34E+5nM ΔG°:  -21.6kJ/mole IC50:  1.25E+5nMpH: 7.0 T: 2°CAssay Description:To test whether GCTs share a common binding pocket on PPA with acarbose, we performed an experiment according to the method of Yonetani and Theorell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM92363(GPESB02)
Affinity DataKi:  3.42E+5nM ΔG°:  -20.6kJ/mole IC50:  1.50E+5nMpH: 7.0 T: 2°CAssay Description:To test whether GCTs share a common binding pocket on PPA with acarbose, we performed an experiment according to the method of Yonetani and Theorell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM92362(GPESB01)
Affinity DataKi:  7.80E+5nM ΔG°:  -18.5kJ/mole IC50:  3.61E+5nMpH: 7.0 T: 2°CAssay Description:To test whether GCTs share a common binding pocket on PPA with acarbose, we performed an experiment according to the method of Yonetani and Theorell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM92364(GPESB07)
Affinity DataKi:  1.01E+6nM ΔG°:  -17.8kJ/mole IC50:  3.56E+5nMpH: 7.0 T: 2°CAssay Description:To test whether GCTs share a common binding pocket on PPA with acarbose, we performed an experiment according to the method of Yonetani and Theorell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120838(CHEMBL1233953)
Affinity DataKi:  1.80E+6nMAssay Description:Inhibition of human pancreatic alpha-amylase assessed as hydrolysis of G3F by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50120841(CHEMBL3616593)
Affinity DataKi: <1.00E+7nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using DP17 amylose as substrate preincubated for 5 mins followed by substrate addition by copper-bicin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50120840(CHEMBL1213470)
Affinity DataKi:  1.80E+7nMAssay Description:Inhibition of human pancreatic alpha-amylase assessed as hydrolysis of G3F by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.5nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  8nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM223316(YPYSCWVRH | piHA-Dm)
Affinity DataIC50:  8.5nMpH: 7.0Assay Description:After kinetic analysis with HPA, piHA-Dm was tested as an inhibitor of ten additional enzymes. The conditions are listed as follows: Agrobacterium fa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataIC50:  10nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50005684(2-Cyclohexyl-2-phenyl-propionic acid 3-diethylamin...)
Affinity DataIC50:  21nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Affinity DataIC50:  46nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50005686(2-Cyclohexyl-2-phenyl-propionic acid 2-diethylamin...)
Affinity DataIC50:  52nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
University Of Canterbury

Curated by ChEMBL
LigandPNGBDBM50005682(2-Cyclohexyl-2-phenyl-propionic acid 4-dimethylami...)
Affinity DataIC50:  190nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Sus scrofa (Pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50568592(CHEMBL4861741)
Affinity DataIC50:  380nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using 1% starch as substrate preincubated for 10 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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