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Found 135 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group D member 1'
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643202(US20240002380, Example 70)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643187(US20240002380, Example 24)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643186(US20240002380, Example 22)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643193(US20240002380, Example 48)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643189(US20240002380, Example 36)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643200(US20240002380, Example 62)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643179(US20240002380, Example 5)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643180(US20240002380, Example 6)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643181(US20240002380, Example 10)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643199(US20240002380, Example 59)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643196(US20240002380, Example 54)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643184(US20240002380, Example 17)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50:  620nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  670nMAssay Description:Agonist activity at Rev-Erbalpha expressed in HEK293 cells coexpressing Gal4 ligand binding domain assessed as inhibition of transcription after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  670nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  710nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50:  790nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643201(US20240002380, Example 68)
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643177(US20240002380, Example 3)
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643183(US20240002380, Example 14)
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643194(US20240002380, Example 49)
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643192(US20240002380, Example 46)
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643182(US20240002380, Example 13)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643198(US20240002380, Example 57)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643191(US20240002380, Example 45)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643185(US20240002380, Example 21)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643197(US20240002380, Example 56)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataKd:  800nMAssay Description:Dissociation constant for binding to REV-ERB-alpha by circular dichroismMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434032(CHEMBL2381195)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434024(CHEMBL2381213)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434027(CHEMBL2381212)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434044(CHEMBL2381194)
Affinity DataEC50:  630nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434023(CHEMBL2380321)
Affinity DataEC50:  630nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434028(CHEMBL2381211)
Affinity DataEC50:  630nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50383684(CHEMBL1961795)
Affinity DataEC50:  500nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434029(CHEMBL2381210)
Affinity DataEC50:  400nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434040(CHEMBL2381207)
Affinity DataEC50:  400nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434043(CHEMBL2381206)
Affinity DataEC50:  400nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434033(CHEMBL2381209)
Affinity DataEC50:  250nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434039(CHEMBL2381193)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434045(CHEMBL2381214)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434037(CHEMBL2381208)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434034(CHEMBL2381205)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434036(CHEMBL2381204)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434035(CHEMBL2381203)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434030(CHEMBL2381202)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434031(CHEMBL2381201)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50434042(CHEMBL2381200)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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