Compile Data Set for Download or QSAR
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Found 672 Enz. Inhib. hit(s) with Target = 'Reverse transcriptase protein'
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50479471(CHEMBL491019 | MK-1107)
Affinity DataKi:  0.220nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50479470(CHEMBL489586 | MK-4965)
Affinity DataKi:  0.390nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50479470(CHEMBL489586 | MK-4965)
Affinity DataKi:  0.390nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484635(CHEMBL1939500)
Affinity DataKi:  0.430nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484496(CHEMBL1928648)
Affinity DataKi:  0.480nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484030(CHEMBL1801256)
Affinity DataKi:  0.5nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484632(Mk-6186 | Mk6186)
Affinity DataKi:  0.580nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484029(CHEMBL1801258)
Affinity DataKi:  0.700nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484045(CHEMBL1801257)
Affinity DataKi:  0.700nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484629(CHEMBL1939503)
Affinity DataKi:  0.940nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484495(CHEMBL1928645)
Affinity DataKi:  1.5nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484493(CHEMBL1928646)
Affinity DataKi:  1.60nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484630(CHEMBL1939502 | MK-7445)
Affinity DataKi:  1.70nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484494(CHEMBL1928647)
Affinity DataKi:  2.10nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484022(CHEMBL1801223)
Affinity DataKi:  2.40nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484031(CHEMBL1801255)
Affinity DataKi:  3.60nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484492(CHEMBL1928643)
Affinity DataKi:  3.70nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484624(CHEMBL1939510)
Affinity DataKi:  3.80nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484040(CHEMBL1801228)
Affinity DataKi:  4.20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484032(CHEMBL1801231)
Affinity DataKi:  4.20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484631(CHEMBL1939501)
Affinity DataKi:  4.30nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484035(CHEMBL1801266)
Affinity DataKi:  4.40nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484024(CHEMBL1801227)
Affinity DataKi:  4.60nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484023(CHEMBL1801230)
Affinity DataKi:  5.20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484634(CHEMBL1939504)
Affinity DataKi:  5.30nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484026(CHEMBL1801225)
Affinity DataKi:  5.5nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  8.5nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484028(CHEMBL1801263)
Affinity DataKi:  9.30nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484033(CHEMBL1801229)
Affinity DataKi:  9.60nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484039(CHEMBL1800087)
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484036(CHEMBL1801265)
Affinity DataKi:  11nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50339536((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...)
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484041(CHEMBL1801254)
Affinity DataKi:  21nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50483329(CHEMBL1650290)
Affinity DataKi:  24nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/T165A mutantMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484633(CHEMBL1939507)
Affinity DataKi:  28nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50339522((+/-)-6-Ethyl-6-[4-[(4-bromophenylthio)methyl]phen...)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484043(CHEMBL1801262)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM2325(2-(cyclopentylsulfanyl)-6-[1-(2,6-difluorophenyl)e...)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  40nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50370476(Combivir | ZIDOVUDINE TRIPHOSPHATE)
Affinity DataKi:  47nMAssay Description:Inhibition of HIV1 reverse transcriptase M41L/D67N/L210W/T215Y mutant by steady state nucleotide incorporation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50164644(2',3'-Dideoxyadenosine Triphosphate (Ddatp) | 2',3...)
Affinity DataKi:  50nMAssay Description:Inhibition of HIV1 reverse transcriptase M41L/D67N/L210W/T215Y mutant by steady state nucleotide incorporation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484038(CHEMBL1801260)
Affinity DataKi:  56nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484497(CHEMBL1928644)
Affinity DataKi:  58nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  65nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484037(CHEMBL1801261)
Affinity DataKi:  69nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50477185(CHEMBL239338)
Affinity DataKi:  80nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50484625(CHEMBL1939509)
Affinity DataKi: >100nMAssay Description:Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50478973(CHEMBL1162283)
Affinity DataKi:  110nMAssay Description:Inhibition of HIV1 reverse transcriptase M41L/D67N/L210W/T215Y mutant by steady state nucleotide incorporation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Merck

Curated by ChEMBL
LigandPNGBDBM50483329(CHEMBL1650290)
Affinity DataKi:  110nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S mutantMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
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