TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 940nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 3.67E+3nMAssay Description:Inhibition of human recombinant PAK2 assessed as phosphorylation of coumarin labeled FRET peptide substrate at Ser/Thr19 preincubated for 10 mins fol...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human PAK2 using RRRLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human PAK2 using RRRLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal 6His-tagged recombinant human PAK2 (3-end residues) expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 12.8nMAssay Description:IC50 values were determined using a 10 concentration point, non-radioactive, functional assay that employs a fluorescence-based, coupled enzyme forma...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human PAK2 by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of PAK2 (unknown origin) using lipid substrate measured after 40 mins by ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of full length PAK2 (unknown origin) by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human PAK2 by radiometric PanQinase activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of PAK2-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of PAK2-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 133nMAssay Description:Inhibition of PAK2-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 244nMAssay Description:Inhibition of PAK2-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Ligand Info
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of PAK2 (unknown origin) using lipid substrate measured after 40 mins by ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild-type human partial length PAK2 (P151 to R525 residues) expressed in bacterial expression system after 1 hr by Z-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAK2 (unknown origin) after 60 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAK2 using ATP as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PAK2 using [KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK] substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Ligand Info
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:Agents: 1-fold kinase buffer without MnCl2: 50 mM HEPES, pH 7.5, 0.0015% Brij-35, 10 mM MgCl2, 2 mM DTT. 1-fold kinase buffer with MnCl2: 50 mM HEPES...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of Pak2 by HTRF kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of Pak2 by HTRF kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 2(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PAK2More data for this Ligand-Target Pair