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Found 161 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PknB'
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279715(CHEMBL4162544)
Affinity DataKi: <1nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279757(CHEMBL4166160)
Affinity DataKi: <1nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279763(CHEMBL4162308)
Affinity DataKi: <1.30nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279744(CHEMBL4165984)
Affinity DataKi: <2nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279743(CHEMBL4170479)
Affinity DataKi:  4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279773(CHEMBL4173915)
Affinity DataKi:  4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279720(CHEMBL4177229)
Affinity DataKi:  5nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279737(CHEMBL4170653)
Affinity DataKi:  6nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279734(CHEMBL4177445)
Affinity DataKi:  13nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279723(CHEMBL4165949)
Affinity DataKi:  15nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279759(CHEMBL4172982)
Affinity DataKi:  17nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279748(CHEMBL4170446)
Affinity DataKi:  23nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279736(CHEMBL4162511)
Affinity DataKi:  23nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279751(CHEMBL4162719)
Affinity DataKi:  24nMAssay Description:Inhibition of human plasma renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279750(CHEMBL4159344)
Affinity DataKi:  29nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279746(CHEMBL4169382)
Affinity DataKi:  38nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279733(CHEMBL4174082)
Affinity DataKi:  40nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279742(CHEMBL4166840)
Affinity DataKi:  46nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279735(CHEMBL4173877)
Affinity DataKi:  50nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279777(CHEMBL4172772)
Affinity DataKi:  60nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279781(CHEMBL4162101)
Affinity DataKi:  72nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279802(CHEMBL4159392)
Affinity DataKi:  81nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279793(CHEMBL4174513)
Affinity DataKi:  82nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279724(CHEMBL4167265)
Affinity DataKi:  88nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279722(CHEMBL4170024)
Affinity DataKi:  98nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279785(CHEMBL4176818)
Affinity DataKi:  150nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279799(CHEMBL4164081)
Affinity DataKi:  150nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279786(CHEMBL4166603)
Affinity DataKi:  150nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279930(CHEMBL4173464)
Affinity DataKi:  190nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279721(CHEMBL4162756)
Affinity DataKi:  230nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279857(CHEMBL4176150)
Affinity DataKi:  310nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279783(CHEMBL4164260)
Affinity DataKi:  310nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279745(CHEMBL4166200)
Affinity DataKi:  960nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279841(CHEMBL4174912)
Affinity DataKi:  990nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279782(CHEMBL4165542)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035670(CHEMBL3338456)
Affinity DataKi:  3.53E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035656(CHEMBL1986389)
Affinity DataKi:  3.86E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50279776(CHEMBL4176789)
Affinity DataKi: >4.00E+3nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035662(CHEMBL3338464)
Affinity DataKi:  5.25E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035666(CHEMBL3338460)
Affinity DataKi:  6.38E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035663(CHEMBL3338463)
Affinity DataKi:  7.01E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035657(CHEMBL3338469)
Affinity DataKi:  7.32E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035658(CHEMBL3338468)
Affinity DataKi:  7.59E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035665(CHEMBL3338461)
Affinity DataKi:  7.68E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035659(CHEMBL3338467)
Affinity DataKi:  9.04E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035664(CHEMBL3338462)
Affinity DataKi:  9.21E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035667(CHEMBL3338459)
Affinity DataKi:  1.08E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035668(CHEMBL3338458)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035661(CHEMBL3338465)
Affinity DataKi:  1.31E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035655(CHEMBL3338470)
Affinity DataKi:  1.85E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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