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Found 117 Enz. Inhib. hit(s) with Target = 'Tau-tubulin kinase 1'
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602886(CHEMBL5182036)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609151(CHEMBL5283456)
Affinity DataIC50:  2.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609143(CHEMBL5268795)
Affinity DataIC50:  2.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609159(CHEMBL5280210)
Affinity DataIC50:  2.70nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609138(CHEMBL5272364)
Affinity DataIC50:  2.80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609144(CHEMBL5279863)
Affinity DataIC50:  7.80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609137(CHEMBL5282072)
Affinity DataIC50:  9.80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609160(CHEMBL5268080)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609145(CHEMBL5271137)
Affinity DataIC50:  18nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609146(CHEMBL5273263)
Affinity DataIC50:  18nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609158(CHEMBL5282902)
Affinity DataIC50:  20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609142(CHEMBL5290581)
Affinity DataIC50:  32nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609157(CHEMBL5274162)
Affinity DataIC50:  37nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609139(CHEMBL5280803)
Affinity DataIC50:  39nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609151(CHEMBL5283456)
Affinity DataIC50:  42nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609141(CHEMBL5288487)
Affinity DataIC50:  57nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609136(CHEMBL5278744)
Affinity DataIC50:  60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609140(CHEMBL5274528)
Affinity DataIC50:  86nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609143(CHEMBL5268795)
Affinity DataIC50:  98nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609137(CHEMBL5282072)
Affinity DataIC50:  114nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602885(CHEMBL5193906)
Affinity DataIC50:  120nMAssay Description:Inhibition of TTBK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50506660(CHEMBL4528881)
Affinity DataIC50:  120nMAssay Description:Inhibition of TTBK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609156(CHEMBL5290252)
Affinity DataIC50:  124nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609144(CHEMBL5279863)
Affinity DataIC50:  164nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609138(CHEMBL5272364)
Affinity DataIC50:  177nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609161(CHEMBL5279159)
Affinity DataIC50:  185nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50429615(CHEMBL2334586)
Affinity DataIC50:  199nMMore data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609158(CHEMBL5282902)
Affinity DataIC50:  224nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609160(CHEMBL5268080)
Affinity DataIC50:  239nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602904(CHEMBL5204869)
Affinity DataIC50:  240nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609146(CHEMBL5273263)
Affinity DataIC50:  259nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609159(CHEMBL5280210)
Affinity DataIC50:  315nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602917(CHEMBL5200069)
Affinity DataIC50:  330nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602907(CHEMBL5193488)
Affinity DataIC50:  340nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609162(CHEMBL5275588)
Affinity DataIC50:  352nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609156(CHEMBL5290252)
Affinity DataIC50:  352nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602930(CHEMBL5181249)
Affinity DataIC50:  360nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602922(CHEMBL5184336)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609162(CHEMBL5275588)
Affinity DataIC50:  377nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602921(CHEMBL5180098)
Affinity DataIC50:  380nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602903(CHEMBL5198544)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602932(CHEMBL5178965)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609152(CHEMBL5272862)
Affinity DataIC50:  414nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602910(CHEMBL5209196)
Affinity DataIC50:  420nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602906(CHEMBL5187459)
Affinity DataIC50:  440nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602920(CHEMBL5187125)
Affinity DataIC50:  450nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602931(CHEMBL5197012)
Affinity DataIC50:  480nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602911(CHEMBL5171328)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602900(CHEMBL5185704 | US11814388, Compound 3)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50609136(CHEMBL5278744)
Affinity DataIC50:  571nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
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