TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Inhibition of 4-methylumbelliferone glucuronidation by human recombinant UGT1A9More data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 3.44E+5nMAssay Description:Drug metabolism assessed as recombinant human UGT1A9 assessed as O-glucuronidation measured as inhibition constant at 10 to 400 uM incubated for 60 m...More data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 5.34E+5nMAssay Description:Substrate inhibition of human recombinant UGT1A9 assessed as IRI-O-5-monoglucuronide formation incubated for 5 mins prior to UDPGA addition measured ...More data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 9.58E+5nMAssay Description:Inhibition of human recombinant UGT1A9 activity expressed in baculovirus-infected Sf9 cellsMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 1.65E+6nMAssay Description:Inhibition of human recombinant UGT1A9 activity expressed in baculovirus-infected Sf9 cellsMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 2.45E+6nMAssay Description:Inhibition of 4-methylumbelliferone glucuronidation by human recombinant UGT1A9More data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of UGT1A9 in human liver microsomes incubated for 30 mins in presence of UDPGA by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of UGT1A9 in human liver microsomes assessed as reduction in mycophenolic acid glucuronidation by tandem mass spectrometry analysisMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of of UGT1A9 in pooled mixed-gender human liver microsomes using 4-methylumbelliferone substrate by HPLC methodMore data for this Ligand-Target Pair