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Found 35 Enz. Inhib. hit(s) with Target = 'Coagulation factor XIII A chain [Q652E]'
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608714(CHEMBL5281897)
Affinity DataIC50:  26nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608719(CHEMBL5269766)
Affinity DataIC50:  29nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50:  100nMMore data for this Ligand-Target Pair
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608720(CHEMBL5285085)
Affinity DataIC50:  102nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM577548(US11472838, Compound Ref. 22)
Affinity DataIC50:  110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608718(CHEMBL5286758)
Affinity DataIC50:  139nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50136842(CHEMBL152117 | GNF-Pf-5230 | N-[2-(4-Hydroxy-pheny...)
Affinity DataIC50:  200nMMore data for this Ligand-Target Pair
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608713(CHEMBL5275210)
Affinity DataIC50:  310nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608710(CHEMBL5290263)
Affinity DataIC50:  350nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608712(CHEMBL5286863)
Affinity DataIC50:  610nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608711(CHEMBL5290280)
Affinity DataIC50:  1.90E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608715(CHEMBL5273935)
Affinity DataIC50:  5.70E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608716(CHEMBL5269322)
Affinity DataIC50:  3.62E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50:  3.70E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608716(CHEMBL5269322)
Affinity DataIC50:  7.63E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50009353(1,5,10-triazadecane | 4-azaoctamethylenediamine | ...)
Affinity DataIC50:  1.00E+5nMMore data for this Ligand-Target Pair
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataIC50:  1.00E+5nMMore data for this Ligand-Target Pair
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185180([2-[[2-(4-tert-Butoxycarbonylpiperazin-1-yl)-2-oxo...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185179(2-(1-Adamantyl)ethyl 4-[2-(prop-2-enoylamino)acety...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185177(1-Adamantylmethyl 4-[2-(prop-2-enoylamino)acetyl]p...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185183(2-(1-Adamantyl)ethyl 4-[2-[(2-bromoacetyl)amino]ac...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185172([2-[[2-[4-(Adamantane-1-carbonyl)piperazin-1-yl]-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185170(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185168([2-[[2-[4-[(4-Methoxycarbonylphenyl)methoxycarbony...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185164((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-(prop-2-...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM60581([2-[[2-[4-[(6-Methoxycarbonyl-2-naphthyl)methoxyca...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185163((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-[(2-brom...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185162(2-Naphthylmethyl 4-[2-(prop-2-enoylamino)acetyl]pi...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185161(Dimethyl-[2-[[2-[4-(2-naphthylmethoxycarbonyl)pipe...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185155([2-[[2-(4-Benzyloxycarbonylpiperazin-1-yl)-2-oxo-e...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM185182([2-[[2-[4-[[5-(Dimethylamino)-1-naphthyl]sulfonyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608717(CHEMBL5273326)
Affinity DataIC50:  1.18E+5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608716(CHEMBL5269322)
Affinity DataKd:  2.53E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails