Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Inhibitory activity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Rattus norvegicus)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMpH: 7.4Assay Description:KI for pyridoxal 5'-phosphate (PLP)-dependent Gamma-amino-N-butyrate transaminase at pH 7.4More data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from bacteriaMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(BOVINE)
Columbia University
Curated by PDSP Ki Database
Columbia University
Curated by PDSP Ki Database
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Rattus norvegicus)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.43E+4nMAssay Description:Activity of GABA transaminase in rat brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Rattus norvegicus)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.10E+4nMAssay Description:Inactivation of GABA-AT in rat brain homogenateMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.10E+4nMAssay Description:Tested for inhibitory activity of the compound against gamma-aminobutyric acid aminotransferase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Reversible inhibition of pig brain GABA-AT using GABA as substrateMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.20E+4nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.30E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.90E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Affinity DataKi: 9.10E+4nMAssay Description:Compound was tested for inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+5nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+5nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.82E+5nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Affinity DataKi: 1.82E+5nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.90E+5nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.90E+5nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.95E+5nMpH: 8.5Assay Description:Compound was tested for inhibitory constant of Gamma-amino-N-butyrate transaminase in pig brain at pH of 8.5 and 25 degree CMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.00E+5nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.30E+5nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.00E+5nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Affinity DataKi: 8.50E+5nMAssay Description:Concentration dependent inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.00E+6nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminase in pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.20E+6nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.30E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.35E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.40E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.59E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.60E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.64E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.00E+6nMpH: 6.5Assay Description:Compound was tested for inhibitory constant of Gamma-amino-N-butyrate transaminase in pig brain at pH of 6.5More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.14E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Affinity DataKi: 2.23E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.27E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+6nMAssay Description:Concentration dependent inactivation of gGamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.40E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.49E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.70E+6nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.80E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.86E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.14E+6nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair