Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.990nMAssay Description:Binding affinity to gastrin releasing peptide receptor (unknown origin)More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonistic activity against cloned human Bombesin receptor bb2 labeled with [125I]- [Tyr] bombesin stably expressed in CHO cells; 0.66-1.3More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair