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Found 16 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group D member 2'
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643181(US20240002380, Example 10)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643199(US20240002380, Example 59)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643191(US20240002380, Example 45)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643190(US20240002380, Example 44)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643178(US20240002380, Example 4)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643177(US20240002380, Example 3)
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50:  560nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  800nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643179(US20240002380, Example 5)
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50095837(CHEMBL3590573)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of REV-ERBbeta (unknown origin) expressed in HEK293 cells incubated for 24 hrs assessed as inhibition of receptor-mediated transcriptional...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643197(US20240002380, Example 56)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643195(US20240002380, Example 51)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643188(US20240002380, Example 34)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643201(US20240002380, Example 68)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM643192(US20240002380, Example 46)
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
Saint Louis University

US Patent
LigandPNGBDBM50095836(CHEMBL3590544)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of REV-ERBbeta (unknown origin) expressed in HEK293 cells incubated for 24 hrs assessed as inhibition of receptor-mediated transcriptional...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed