Affinity DataKi: 60nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.19E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.91E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.24E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.59E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.02E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.88E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.37E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.77E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of PKN1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of PRK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of PKN1 (unknown origin) incubated for 1 hr by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human PKN1 using KKLNRTLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human PKN1 using KKLNRTLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of full-length recombinant human GST-tagged PKN1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of PKN1 using ATP as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 547nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PKN-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Protein kinase C related kinase 1 (PRK1)More data for this Ligand-Target Pair