TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 32nM ΔG°: -43.5kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 48nM ΔG°: -42.5kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 67nM ΔG°: -41.6kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 275nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 310nM ΔG°: -37.8kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 360nM ΔG°: -37.4kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 840nM ΔG°: -35.3kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 942nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataKi: 5.84E+3nM ΔG°: -30.4kJ/molepH: 6.8 T: 2°CAssay Description:AANAT activity was measured using a spectrophotometric assay in which the enzymatic product CoASH concentration were determined indirectly by monitor...More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.99E+4nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 7.12E+4nMAssay Description:Inhibition of serotonin N-acetyl-transferaseMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 180nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 390nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 610nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 680nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 700nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 1.43E+3nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 3.78E+3nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of ovine AANAT by TLC-based radioactive assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of ovine AANAT by TLC-based radioactive assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.52E+4nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.84E+4nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.99E+4nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Homo sapiens (Human))
Johns Hopkins University School Of Medicine
Johns Hopkins University School Of Medicine
Affinity DataIC50: 4.00E+4nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.52E+4nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.29E+4nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair
TargetSerotonin N-acetyltransferase(Ovis aries)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.02E+5nMAssay Description:Inhibition of ovine AANAT by spectrophotometric assayMore data for this Ligand-Target Pair