Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Short transient receptor potential channel 1/4'
TargetShort transient receptor potential channel 1/4(Homo sapiens)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50519465(CHEMBL4466522)
Affinity DataIC50:  0.0330nMAssay Description:Inhibition of human TRPC4/human TRPC1 expressed in HEK293 cells assessed as reduction in englerin A-induced calcium entry incubated for 30 mins by Fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetShort transient receptor potential channel 1/4(Homo sapiens)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50519489(CHEMBL4450705)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at TRPC4/TRPC1 in human A498 cells assessed as reduction in englerin A-induced calcium entry preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed