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Found 200 Enz. Inhib. hit(s) with Target = 'Transcriptional enhancer factor TEF-3'
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataKi:  2.60E+3nMAssay Description:Reversible inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Codon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547126(CHEMBL4763473)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50604885(CHEMBL5177177)
Affinity DataKi: >4.00E+5nMAssay Description:Displacement of FAM- labeled YAP1 peptide from TEAD4 (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as inhi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50535723(CHEMBL4567546)
Affinity DataIC50:  9nMAssay Description:Inhibition of human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) interaction with N-biotinylated YAP (60 to 100 residues) inc...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626331(US11787775, Compound 16-C)
Affinity DataIC50:  10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626350(2-[[[4-cyano-7-(4-isopropyl-2- thienyl)-2,3-dihyd...)
Affinity DataIC50:  10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626350(2-[[[4-cyano-7-(4-isopropyl-2- thienyl)-2,3-dihyd...)
Affinity DataIC50:  10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50535722(CHEMBL4468725)
Affinity DataIC50:  16nMAssay Description:Inhibition of human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) interaction with N-biotinylated YAP (60 to 100 residues) inc...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626336(2-[[[4-fluoro-7-(4-isopropylphenyl)- 2,3-dihydrob...)
Affinity DataIC50:  20nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626335(2-[[[4-(4-isopropylphenyl)-6,7- dihydrofuro[3,2-d...)
Affinity DataIC50:  20nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626323(US11787775, Compound 8 | methyl 2-[[[4-cyano-7-(4-...)
Affinity DataIC50:  20nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626318(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  20nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626318(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  20nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626318(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  30nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626342(2-[[[4-cyano-7-(2-fluoro-4- isopropyl-phenyl)-2,3...)
Affinity DataIC50:  30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626333(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)
Affinity DataIC50:  30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626332(US11787775, Compound 16-D)
Affinity DataIC50:  30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626317(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)
Affinity DataIC50:  30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626358(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)
Affinity DataIC50:  40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626324(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626326(7-(4-isopropylphenyl)-5-[(2- methylene-3-oxo-buty...)
Affinity DataIC50:  40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626316(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)
Affinity DataIC50:  40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50535724(CHEMBL4467555)
Affinity DataIC50:  45nMAssay Description:Inhibition of human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) interaction with N-biotinylated YAP (60 to 100 residues) inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626354(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)
Affinity DataIC50:  50nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626337(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrofu...)
Affinity DataIC50:  50nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50535715(CHEMBL4476332)
Affinity DataIC50:  56nMAssay Description:Inhibition of human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) interaction with N-biotinylated YAP (60 to 100 residues) inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626362(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)
Affinity DataIC50:  60nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626365(2-[[[7-cyano-4-[4-(pentafluoro- lambda6-sulfanyl)...)
Affinity DataIC50:  60nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626354(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)
Affinity DataIC50:  60nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  70nMAssay Description:Binding affinity to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626319(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  80nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626361(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)
Affinity DataIC50:  80nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626358(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)
Affinity DataIC50:  80nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626355(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)
Affinity DataIC50:  80nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626319(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  80nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626364(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)
Affinity DataIC50:  90nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547134(CHEMBL4787565)
Affinity DataIC50:  100nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM626324(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  100nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626330(2-[[[4-cyano-7-[4- (trifluoromethyl)phenyl]-2,3- ...)
Affinity DataIC50:  110nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626334(2-[[[4-cyano-7-[4-(1,1- difluoroethyl)phenyl]-2,3...)
Affinity DataIC50:  110nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626324(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  120nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626361(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)
Affinity DataIC50:  120nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626339(2-[[[6-methoxy-5-[(E)-2-[trans-4- (trifluoromethy...)
Affinity DataIC50:  140nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626354(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)
Affinity DataIC50:  140nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626360(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)
Affinity DataIC50:  140nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626322(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataIC50:  160nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626355(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)
Affinity DataIC50:  160nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626347(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)
Affinity DataIC50:  170nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM626328(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)
Affinity DataIC50:  180nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM626354(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)
Affinity DataIC50:  180nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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