TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 48.7nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 55.4nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 75.9nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 85.5nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 88.6nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 105nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 222nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 354nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 553nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 905nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against Calpain IMore data for this Ligand-Target Pair