Affinity DataEC50: 5.40E+3nMAssay Description:Agonist activity at recombinant GluA2 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 5.40E+3nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 2 (GluR2) using rat cort...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Mus musculus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.40E+4nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Metabotropic glutamate receptor 1 using rat cortical slice ...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rattus norvegicus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 3.80E+4nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 4 (GluR4) using rat cort...More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+5nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 3 (GluR3) using rat cort...More data for this Ligand-Target Pair
Affinity DataEC50: 2.02E+5nMAssay Description:Agonist activity at recombinant GluA3 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.02E+5nMAssay Description:Agonist activity at recombinant GluA3 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair