Found 30 of ec50 for monomerid = 50029051 
Affinity DataEC50: 5.5nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP levels by DELFIA methodMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Agonist activity at human adrenergic beta3 receptor expressed in CHO cells assessed as [3H]cAMP levels by radiolabeled ligand based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Agonist activity at human alpha1A-adrenergic receptor expressed in HEK293 cells assessed as calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:In vitro agonist potency towards Alpha-1D adrenergic receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Effective concentration for Beta-1 adrenergic receptor mediated inhibition of neurotransmission in field-stimulated reserpine pretreated guinea pig i...More data for this Ligand-Target Pair
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonistic potency at human adrenergic alpha-2B receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonist activity at human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 118nMAssay Description:Agonist activity at human adrenoceptor alpha2A expressed in CHOK1 cells assessed as stimulation of agonist-induced [35S]GTPgammaS binding by scintill...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 129nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO-K1 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 213nMAssay Description:Activity for Beta-2 adrenergic receptor was assessed from effect on relaxation of guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Agonistic potency at beta-1 adrenergic receptor for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonist activity at human recombinant adrenergic alpha2A receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonistic potency at human adrenergic alpha-2A receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonist activity at human adrenergic alpha-2A receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonist activity at human adrenergic alpha-2C receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita Degli Studi Di Camerino
Curated by ChEMBL
Universita Degli Studi Di Camerino
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.18E+3nMAssay Description:In vitro agonist potency towards Alpha-1A adrenergic receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetBeta-3 adrenergic receptor(Rattus norvegicus)
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Effective dose for contraction of reserpine-pretreated rat vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+3nMAssay Description:In vitro agonist potency towards Alpha-1A adrenergic receptor in canine prostateMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Effective dose required to stimulate contractions in isolated guinea pig atrium.More data for this Ligand-Target Pair
Affinity DataEC50: 1.02E+4nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
TargetBeta-3 adrenergic receptor(Rattus norvegicus)
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.00E+5nMAssay Description:Activity for beta 3-adrenoceptor was assessed from effect on stimulation of lipolysis in rat adipocytes.More data for this Ligand-Target Pair
