Affinity DataEC50: 0.400nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 391nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >6.50E+3nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair