Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ec50 for monomerid = 50276073
TargetHistamine H3 receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50276073(CHEMBL502339 | N1-[3-(1H-Imidazol-4-yl)propyl]-N2-...)
Affinity DataEC50:  1.64nMAssay Description:Activity at human recombinant histamine H3 receptor expressed in Sf9 cells coexpressing Galphai, G-beta-1-gamma-2 and RGS4 by steady-state GTPase act...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50276073(CHEMBL502339 | N1-[3-(1H-Imidazol-4-yl)propyl]-N2-...)
Affinity DataEC50:  6.30nMAssay Description:Activity at human recombinant histamine H4 receptor-RGS4 fusion protein expressed in Sf9 cells coexpressing Galphai2 and G-beta-1-gamma-2 by steady-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50276073(CHEMBL502339 | N1-[3-(1H-Imidazol-4-yl)propyl]-N2-...)
Affinity DataEC50:  21nMAssay Description:Activity at guinea pig recombinant histamine H2 receptor-Gsalpha fusion protein expressed in Sf9 cells by steady-state GTPase activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50276073(CHEMBL502339 | N1-[3-(1H-Imidazol-4-yl)propyl]-N2-...)
Affinity DataEC50:  38.0nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig spontaneously beating right atrium assessed as positive chronotropic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50276073(CHEMBL502339 | N1-[3-(1H-Imidazol-4-yl)propyl]-N2-...)
Affinity DataEC50:  109nMAssay Description:Activity at human recombinant histamine H2 receptor-Gsalpha fusion protein expressed in Sf9 cells by steady-state GTPase activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed