Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ec50 for monomerid = 50428095
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50428095(CHEMBL2331646)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human TGR5 expressed in deoxycycline-induced Flp-In-CHO-TO cells assessed as increase in intracellular cAMP measured after 48 hrs...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50428095(CHEMBL2331646)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human TGR5 expressed in uninduced Flp-In-CHO-TO cells assessed as increase in intracellular cAMP measured after 48 hrs by HTRF co...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50428095(CHEMBL2331646)
Affinity DataEC50:  3.93E+3nMAssay Description:Agonist activity at rat TGR5 expressed in deoxycycline-induced CHO cells assessed as increase in intracellular cAMP measured after 48 hrs by HTRF com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50428095(CHEMBL2331646)
Affinity DataEC50:  5.62E+3nMAssay Description:Agonist activity at mouse TGR5 expressed in deoxycycline-induced CHO cells assessed as increase in intracellular cAMP measured after 48 hrs by HTRF c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed