TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at alpha4beta 2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 7.30nMAssay Description:In vitro binding affinity by inhibiting [3H]dopamine release in rat brain tissue at Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 77nMAssay Description:Agonist activity at alpha4beta2 nAChR in rat frontal cortex membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in SH-EP1 cells assessed as 86Rb+ ion efflux after 9.5 mins by flip-plate techniqueMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Agonist activity at human alpha4beta2 nACHR expressed in human SHEP1 cells assessed as stimulation of 86Rb+ ion efflux after 5 mins by liquid scintil...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in human SH-EP1 cells assessed as increase of carbamylcholine-induced 86Rb+ ion efflux by liqui...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 295nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in human SH-EP1 cells assessed as stimulation of 86Rb+ efflux preincubated for 10 mins by liqui...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 295nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in human SH-EP1 cells assessed as stimulation of 86Rb+ efflux preincubated for 10 mins by liqui...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at human nAChR alpha4beta2 in human SH-EP1 cells assessed as induction in rubidium effluxMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Compound was evaluated for functional potencies and efficacies at human Nicotinic acetylcholine receptor subtype TE671 (muscle)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 591nMAssay Description:Agonist activity at alpha4beta2 nAChR in rat thalamic synaptosomes assessed as increase in 86Rb effluxMore data for this Ligand-Target Pair
Affinity DataEC50: 720nMAssay Description:Agonist activity at mouse neuronal acetylcholine receptor subunit alpha4beta2 expressed in HEK293T cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 724nMAssay Description:Agonist activity at mouse neuronal acetylcholine receptor subunit alpha4beta2 expressed in HEK293T cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 740nMpH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ul of 0.2 mg/ml an...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Agonist activity at human brain alpha4beta2 nAChR expressed in CHO cells by patch clamp electrophysiological assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration against rat alpha4-beta2 nicotinic acetylcholinereceptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 1.07E+3nMAssay Description:Agonist activity at rat alpha7 nAchR expressed in rat GH4C1 cells assessed as stimulation of calcium flux by FLIPRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at rat alpha-7 nAChR expressed in GH4C1-F7 cells assessed as effect on calcium influx by FLIPRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Iqm-Csic
Curated by ChEMBL
Iqm-Csic
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Iqm-Csic
Curated by ChEMBL
Iqm-Csic
Curated by ChEMBL
Affinity DataEC50: 1.51E+3nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+3nMAssay Description:Agonist activity at human recombinant alpha7 nAChR expressed in rat GH3 cells by calcium influx assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:The functional properties of the ligands were determined by 86Rb+ efflux assays in cells expressing α3β4 and α4β2 nAChR subtypes....More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Agonist activity at human alpha4beta2 nAChR assessed as stimulation of [86Rb+] efflux after 2 mins by cell-based liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Agonist activity at human alpha4beta2 nACHR expressed in HEK293 cells assessed as stimulation of 86Rb+ efflux after 2 hrs by liquid scintillation cou...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at alpha4beta2 nACHR in human SHEP1 cell membranes assessed as stimulation of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at alpha4beta2 nAChR in human SH-EP1 cells assessed as calcium flux by calcium4-based FLIPR assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Compound was evaluated for functional potencies and efficacies at human Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Compound was evaluated for functional potencies and efficacies at rat Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataEC50: 4.30E+3nMAssay Description:Agonistic potency against nicotinic acetylcholine receptor alpha3-beta4More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Agonist activity at human recombinant alpha4beta2 nAChR expressed in human IMR32 cells assessed as calcium dynamics by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.71E+3nMAssay Description:Agonist activity at human alpha7 nAChR expressed in mouse Neuro2a cells co-expressing chaperone NACHO assessed as increase in intracellular Ca2+ leve...More data for this Ligand-Target Pair
Affinity DataEC50: 4.71E+3nMAssay Description:Agonist activity at human alpha7 nAChR expressed in mouse Neuro2a cells co-expressing chaperone NACHO assessed as increase in intracellular Ca2+ leve...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Tested for functional activity against neuronal nicotinic acetylcholine receptor(nAChR) expressed in K177 cells using isotopic rubidium efflux assay.More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Binding affinity towards nAChR (alpha4-beta2) by the displacement of [3H]-(-)-cytisine in whole rat brain membranes.More data for this Ligand-Target Pair
TargetResistance to inhibitors of cholinesterase protein 3(Pig roundworm)
Iowa State University Research Foundation
US Patent
Iowa State University Research Foundation
US Patent
Affinity DataEC50: 6.21E+3nMAssay Description:Nematode eggs are isolated from fresh feces by centrifugation and flotation. The eggs are washed and inspected to confirm embryonation has not starte...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataEC50: 6.60E+3nMAssay Description:Agonist activity at human recombinant alpha4beta2 nicotinic acetylcholine receptor expressed in HEK293 cells assessed as changes in intracellular cal...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 6.60E+3nMAssay Description:Agonist activity at recombinant human alpha-4-beta-2 nAChR expressed in HEK293 cells assessed as induction of calcium influx by FLIPR assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
Sibia Neurosciences
Curated by PDSP Ki Database
Sibia Neurosciences
Curated by PDSP Ki Database
Affinity DataEC50: 7.10E+3nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataEC50: 9.40E+3nMAssay Description:Agonist activity at human recombinant alpha3beta4 nAChR expressed in human IMR32 cells assessed as calcium dynamics by FLIPR assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Berne
Curated by ChEMBL
University Of Berne
Curated by ChEMBL
Affinity DataEC50: 9.40E+3nMAssay Description:Agonist activity at alpha-4-beta-2 in IMR-32cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at rat alpha-4-beta-2 nACHR by rubidium efflux assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
Sibia Neurosciences
Curated by PDSP Ki Database
Sibia Neurosciences
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+4nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Mus musculus)
University Of Hull
Curated by ChEMBL
University Of Hull
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at mouse TRPA1 expressed in CHO cells assessed as increase in calcium influx by patch clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 1.30E+4nMAssay Description:Effective concentration against rat alpha7 nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 1.40E+4nMAssay Description:Agonist activity at rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:Activation of TRPA1 channelMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataEC50: 1.90E+4nMAssay Description:Agonist activity at rat brain alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
University Of Wollongong
Curated by ChEMBL
University Of Wollongong
Curated by ChEMBL
Affinity DataEC50: 1.98E+4nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Compound was evaluated for functional potencies and efficacies at rat Nicotinic acetylcholine receptor subtype PC12 (ganglionic)More data for this Ligand-Target Pair